SCHEMBL8314940

SCHEMBL8314940

CN(c1ncc2ncnc(Nc3ccc(Cl)c(Cl)c3)c2n1)[C@H]1CC[C@H](O)CC1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EGFR P00533 9/20 0.48
ERBB2 P04626 4/20 0.47
HPGD P15428 1/20 0.47
HTT P42858 1/20 0.47
MAPT P10636 1/20 0.44
BRAF P15056 8/20 0.43
EPHA2 P29317 3/20 0.40
KDR P35968 3/20 0.40
EPHB4 P54760 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8314944 1.00 EGFR (0.48) EGFRERBB2HPGDHTTMAPT
SCHEMBL8316549 0.92 EGFR (0.58) EGFRERBB2HPGDHTTMAPT
SCHEMBL8316553 0.92 EGFR (0.58) EGFRERBB2HPGDHTTMAPT
SCHEMBL8319415 0.88 EGFR (0.54) EGFRERBB2HPGDHTTBRAF
SCHEMBL8319409 0.88 EGFR (0.54) EGFRERBB2HPGDHTTBRAF
SCHEMBL8316432 0.85 EGFR (0.69) EGFRERBB2HTTBRAF
SCHEMBL8316426 0.85 EGFR (0.69) EGFRERBB2HTTBRAF
SCHEMBL8316033 0.84 EGFR (0.70) EGFR
SCHEMBL8316029 0.84 EGFR (0.70) EGFR
SCHEMBL6996564 0.82 EGFR (0.58) EGFRERBB2HPGDHTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed