SCHEMBL8315008

SCHEMBL8315008

CNc1ncc2ncnc(Nc3cccc(C)c3)c2n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EGFR P00533 18/20 1.00
ERBB2 P04626 2/20 0.57
HTT P42858 1/20 0.54
HIF1A Q16665 1/20 0.54
MAPK1 P28482 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8316963 0.92 EGFR (0.86) EGFRERBB2HTTHIF1AMAPK1
SCHEMBL8316429 0.89 EGFR (0.80) EGFRERBB2HTTHIF1AMAPK1
SCHEMBL8317851 0.87 EGFR (0.77) EGFRERBB2HTTHIF1A
SCHEMBL8318090 0.87 EGFR (0.77) EGFRHTTHIF1A
SCHEMBL8317470 0.87 EGFR (0.77) EGFRHTTHIF1A
SCHEMBL8318451 0.87 EGFR (0.77) EGFRHTTHIF1A
SCHEMBL8319428 0.85 EGFR (0.73) EGFRERBB2HTTHIF1AMAPK1
SCHEMBL8317938 0.85 EGFR (0.73) EGFRHTTHIF1A
SCHEMBL8316727 0.85 EGFR (0.73) EGFRERBB2HTTHIF1A
SCHEMBL8320643 0.84 EGFR (0.72) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed