SCHEMBL8315248

SCHEMBL8315248

COC(=O)/C=C/c1cccc(Br)c1.C[Si](C)(C)Cl

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B3 P37058 1/20 0.58
PKM P14618 1/20 0.56
SLC6A19 Q695T7 1/20 0.55
MEN1 O00255 3/20 0.52
KMT2A Q03164 3/20 0.52
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52
MAOB P27338 2/20 0.51
BACE1 P56817 1/20 0.51
MAOA P21397 1/20 0.51
POLB P06746 1/20 0.51
TTR P02766 1/20 0.50
APP P05067 1/20 0.50
HTT P42858 1/20 0.49
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
PTPN1 P18031 1/20 0.48
CYP2D6 P10635 1/20 0.47
CYP1B1 Q16678 1/20 0.47
EPHX2 P34913 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8315251 1.00 HSD17B3 (0.58) HSD17B3PKMSLC6A19MEN1KMT2A
SCHEMBL322249 0.93 HSD17B3 (0.67) HSD17B3PKMSLC6A19MEN1KMT2A
SCHEMBL1132527 0.93 HSD17B3 (0.67) HSD17B3PKMSLC6A19MEN1KMT2A
SCHEMBL69618 0.81 TTR (0.66) MEN1KMT2ATTRAPPHTT
SCHEMBL29247898 0.78 HSD17B3 (0.73) HSD17B3PKMSLC6A19KMT2AMAOB
SCHEMBL1105481 0.78 HSD17B3 (0.73) HSD17B3PKMSLC6A19KMT2AMAOB
SCHEMBL30963011 0.78 HSD17B3 (0.73) HSD17B3PKMSLC6A19KMT2AMAOB
SCHEMBL17157974 0.78 HSD17B3 (0.63) HSD17B3PKMSLC6A19MEN1KMT2A
SCHEMBL17157975 0.78 HSD17B3 (0.63) HSD17B3PKMSLC6A19MEN1KMT2A
SCHEMBL2500242 0.77 CYP1A2 (0.67) MEN1KMT2ANPC1RAB9AMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0892784-A1 AMINOISOQUINOLINES AND AMINOTHIENOPYRIDINE DERIVATIVES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS Astra Pharmaceuticals Limited (GB) 1999-01-27 EP disclosed
WO-1997038977-A1 AMINOISOQUINOLINES AND AMINOTHIENOPYRIDINE DERIVATIVES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS ASTRA PHARMACEUTICALS LTD. (GB) 1997-10-23 WO disclosed