SCHEMBL8315843

SCHEMBL8315843

COc1cc2c(cc1OC)C(O)(c1cccc[n+]1[O-])CC(C)(C)CO2

nearest known ligand 0.32

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.32
KDM4E B2RXH2 2/20 0.31
LMNA P02545 2/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP3A4 P08684 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
MAPK1 P28482 1/20 0.31
HSD17B10 Q99714 1/20 0.31
FTO Q9C0B1 1/20 0.30
HTT P42858 1/20 0.30
MT-ND4 P03905 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8315522 0.86 BACE1 (0.33) SCN9AKDM4ELMNAALDH1A1CYP3A4
SCHEMBL8311155 0.85 AKR1B1 (0.32)
SCHEMBL8314858 0.83
SCHEMBL8310355 0.82 AKR1B1 (0.34)
SCHEMBL8311440 0.82 AKR1B1 (0.34)
SCHEMBL8315240 0.81
SCHEMBL8315596 0.81 MAP3K14 (0.34) LMNAALDH1A1
SCHEMBL8315276 0.81 BACE1 (0.33)
SCHEMBL8313605 0.80 HTR2B (0.35)
SCHEMBL8313650 0.80 PDK2 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP disclosed
US-5652252-A POTASSIUM CHANNEL ACTIVATORS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-07-29 US disclosed
US-5602152-A POTASSIUM CHANNEL MODULATOR MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-02-11 US disclosed
EP-0626954-A1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GmbH (DE) 1994-12-07 EP disclosed
WO-1994013658-A2 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1994-06-23 WO disclosed