SCHEMBL8317118

SCHEMBL8317118

COc1ccc2c(C3CCNCC3)c[nH]c2c1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 5/20 0.57
ADRB2 P07550 1/20 0.57
APP P05067 5/20 0.56
HTR6 P50406 2/20 0.48
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
MAPT P10636 1/20 0.48
HTR4 Q13639 1/20 0.47
HTR2A P28223 2/20 0.47
HTR2B P41595 1/20 0.47
MTNR1A P48039 1/20 0.46
MTNR1B P49286 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11841895 0.99 HTR2C (0.58) HTR2CADRB2APPHTR6KDM4E
SCHEMBL2264043 0.89 HTR2C (0.60) HTR2CADRB2APPHTR6HTR4
Hydrochloric Acid SCHEMBL11847902 0.87 HTR2C (0.59) HTR2CADRB2APPHTR6KDM4E
SCHEMBL4676883 0.81 HTR2C (0.62) HTR2CADRB2APPHTR2A
SCHEMBL25079811 0.81 HTR2C (0.58) HTR2CADRB2APPHTR6MAPT
SCHEMBL6358819 0.81 HTR2C (0.58) HTR2CADRB2APPHTR6MAPT
SCHEMBL25079814 0.81 HTR2C (0.58) HTR2CADRB2APPHTR6MAPT
SCHEMBL26776434 0.79 HTR2A (0.46) HTR2CAPPHTR6KDM4EALDH1A1
SCHEMBL26776464 0.79 HTR2A (0.46) HTR2CAPPHTR6KDM4EALDH1A1
SCHEMBL16801567 0.78 HTR2C (0.56) HTR2CADRB2APPKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3993764-A 3-(4*-PIPERIDYL)-INDOLES ROUSSEL-UCLAF (FR) 1976-11-23 US claimed
EP-0536419-B1 TRICYCLIC TRIAZOLE DERIVATIVES, PRODUCTION AND USE THEREOF TORAY INDUSTRIES (JP) 1999-10-13 EP disclosed
US-5683998-A ANTIINFLAMMATORY AGENTS, ANTIALLERGENS, ANTIPAF AGENTS TORAY INDUSTRIES, INC. (JP) 1997-11-04 US disclosed
US-5670511-A Indolepiperidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-09-23 US disclosed
EP-0722942-A1 Indole piperidine derivatives MERCK PATENT GmbH (DE) 1996-07-24 EP disclosed
EP-0536419-A1 TRICYCLIC TRIAZOLE DERIVATIVE, PRODUCTION THEREOF, AND USE THEREOF TORAY INDUSTRIES, INC. (JP) 1993-04-14 EP disclosed
US-3993764-A 3-(4*-PIPERIDYL)-INDOLES ROUSSEL-UCLAF (FR) 1976-11-23 US disclosed
US-3947578-A Omega-[4-(3\"-indolyl)-piperidino]-alkyl-arylketones as nevroleptics ROUSSEL UCLAF (FR) 1976-03-30 US disclosed