SCHEMBL8319581

SCHEMBL8319581

CCOC(=O)c1cccc(Nc2ncnc3cnc(NC4CC4)nc23)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
LMNA P02545 2/20 0.58
POLB P06746 1/20 0.58
HPGD P15428 3/20 0.57
BRAF P15056 4/20 0.52
EGFR P00533 3/20 0.50
KDM4E B2RXH2 1/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
MAPKAPK2 P49137 1/20 0.50
ERBB2 P04626 1/20 0.49
HTT P42858 1/20 0.49
TP53 P04637 4/20 0.48
CSNK2A1 P68400 4/20 0.47
THRB P10828 1/20 0.46
CSNK2A2 P19784 3/20 0.46
CSNK2B P67870 3/20 0.46
ALDH1A1 P00352 1/20 0.46
CSNK2A3 Q8NEV1 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7580907 0.84 EGFR (0.55) HPGDBRAFEGFRERBB2HTT
SCHEMBL8318379 0.83 EGFR (0.55) HPGDBRAFEGFRERBB2HTT
SCHEMBL8313532 0.83 EGFR (0.56) MAPTSMN1; SMN2LMNAHPGDBRAF
SCHEMBL7581241 0.82 EGFR (0.55) HPGDBRAFEGFRERBB2HTT
SCHEMBL7577862 0.82 CSNK2A1 (0.51) HPGDBRAFEGFRERBB2HTT
SCHEMBL8319428 0.82 EGFR (0.73) HPGDBRAFEGFRERBB2HTT
SCHEMBL8314008 0.80 EGFR (0.60) HPGDBRAFEGFRERBB2HTT
SCHEMBL8314004 0.80 EGFR (0.60) HPGDBRAFEGFRERBB2HTT
SCHEMBL8318922 0.80 EGFR (0.62) HPGDBRAFEGFRERBB2HTT
SCHEMBL8318928 0.80 EGFR (0.62) HPGDBRAFEGFRERBB2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed