SCHEMBL8319640

SCHEMBL8319640

O=C(O)/C=C/c1ccc(Cn2cnc3ccccc32)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.63
HDAC8 Q9BY41 1/20 0.63
CYP11B1 P15538 7/20 0.62
CYP11B2 P19099 7/20 0.62
TNF P01375 1/20 0.62
HDAC6 Q9UBN7 1/20 0.62
HTT P42858 4/20 0.58
SMN1; SMN2 Q16637 4/20 0.58
MAPK1 P28482 1/20 0.58
LMNA P02545 5/20 0.57
CYP1A2 P05177 2/20 0.51
TBXAS1 P24557 2/20 0.51
USP2 O75604 1/20 0.51
MEN1 O00255 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C19 P33261 1/20 0.51
KMT2A Q03164 1/20 0.51
TSHR P16473 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3969678 0.82 CYP11B1 (0.71) HDAC1HDAC8CYP11B1CYP11B2TNF
SCHEMBL13907295 0.80 CYP11B1 (0.89) HDAC1CYP11B1CYP11B2TNFHDAC6
SCHEMBL1750364 0.80 HDAC1 (0.73) HDAC1CYP11B1CYP11B2TNFHDAC6
SCHEMBL230002 0.79 CYP11B1 (1.00) HDAC1CYP11B1CYP11B2TNFHDAC6
SCHEMBL31357411 0.79 CYP11B1 (1.00) HDAC1CYP11B1CYP11B2TNFHDAC6
SCHEMBL17942160 0.78 CYP11B1 (0.69) HDAC1CYP11B1CYP11B2TNFHDAC6
SCHEMBL3368462 0.77 HDAC1 (1.00) HDAC1HDAC8HDAC6
SCHEMBL3368458 0.77 HDAC1 (1.00) HDAC1HDAC8HDAC6
SCHEMBL12850040 0.76 HDAC6 (1.00) HDAC1HDAC8CYP11B1CYP11B2TNF
SCHEMBL7672864 0.76 CYP11B1 (0.75) HDAC1CYP11B1CYP11B2TNFHDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004063169-A1 HYDROXAMID ACID DERIVATIVES AS HISTONE DEACETYLASE (HDAC) INHIBITORS ASTELLAS PHARMA INC. (JP) 2004-07-29 WO disclosed