SCHEMBL8319904

SCHEMBL8319904

CSc1cccc(Oc2ncc(F)cc2C(=O)N[C@H]2CC[C@@H](NC(=O)c3cc(Oc4ccccc4)cc(Oc4ccccc4)c3)CC2)c1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.51
PDE4B Q07343 17/20 0.51
PDE4A P27815 1/20 0.51
PDE4D Q08499 1/20 0.51
PKM P14618 1/20 0.47
PTGER4 P35408 1/20 0.46
CYP3A4 P08684 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5813532 1.00 NPC1 (0.51) NPC1PDE4BPDE4APDE4DPKM
SCHEMBL5839255 0.92 PDE4B (0.51) PDE4BPDE4APDE4DPTGER4CYP3A4
SCHEMBL8312818 0.90 PDE4B (0.54) PDE4BPDE4APDE4DCYP3A4
SCHEMBL5840103 0.90 PDE4B (0.54) PDE4BPDE4APDE4DCYP3A4
SCHEMBL5839406 0.88 PDE4B (0.55) PDE4BPDE4APDE4DCYP3A4
SCHEMBL5839482 0.88 PDE4B (0.52) PDE4BPDE4APDE4DPTGER4CYP3A4
SCHEMBL8313200 0.88 PDE4B (0.54) PDE4BPDE4APDE4DPTGER4CYP3A4
SCHEMBL5839644 0.88 PDE4B (0.54) PDE4BPDE4APDE4DPTGER4CYP3A4
SCHEMBL5839648 0.88 PDE4B (0.54) PDE4BPDE4APDE4DPTGER4CYP3A4
SCHEMBL8315195 0.88 PDE4B (0.51) PDE4BPDE4APDE4DCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005009966-A1 NICOTINAMIDE DERIVATIVES USEFUL AS PDE4 INHIBITORS PFIZER LIMITED (GB) 2005-02-03 WO disclosed