SCHEMBL8320082

SCHEMBL8320082

COc1ccc(Nc2ncnc3cnc(NC4CC4)nc23)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 6/20 0.56
HTT P42858 2/20 0.56
ERBB2 P04626 1/20 0.56
HPGD P15428 1/20 0.56
MERTK Q12866 2/20 0.52
SYK P43405 2/20 0.49
MAPT P10636 1/20 0.48
GRM1 Q13255 1/20 0.48
BRAF P15056 1/20 0.48
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
SHMT2 P34897 1/20 0.47
LCK P06239 2/20 0.46
PDPK1 O15530 1/20 0.46
MAPK6 Q16659 1/20 0.46
IRAK4 Q9NWZ3 1/20 0.46
NCOA1 Q15788 1/20 0.46
NCOA3 Q9Y6Q9 1/20 0.46
AURKA O14965 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8319961 0.87 EGFR (0.58) EGFRHTTERBB2HPGDSYK
SCHEMBL8312571 0.87 CSNK2A1 (0.60) EGFRHTTERBB2HPGDMERTK
SCHEMBL8315463 0.85 EGFR (0.61) EGFRHTTERBB2HPGDMERTK
SCHEMBL8318401 0.85 EGFR (0.56) EGFRHTTERBB2HPGDBRAF
SCHEMBL8321212 0.85 EGFR (0.64) EGFRHTTERBB2HPGDSYK
SCHEMBL8315669 0.84 EGFR (0.56) EGFRHTTERBB2HPGDBRAF
SCHEMBL23538175 0.83 EGFR (0.53) EGFRERBB2
SCHEMBL6999398 0.82 SYK (0.53) EGFRHTTERBB2HPGDMERTK
SCHEMBL6999389 0.82 SYK (0.53) EGFRHTTERBB2HPGDMERTK
SCHEMBL8317471 0.82 EGFR (0.61) EGFRHTTERBB2HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed