SCHEMBL8320538

SCHEMBL8320538

CCCCOc1ncc2ncnc(Nc3cccc(C)c3)c2n1

nearest known ligand 0.64

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EGFR P00533 16/20 0.64
HTT P42858 1/20 0.51
HIF1A Q16665 1/20 0.51
MAPK1 P28482 1/20 0.49
ERBB2 P04626 1/20 0.49
SYK P43405 1/20 0.48
AURKB Q96GD4 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8318245 0.85 EGFR (0.77) EGFRHTTHIF1AMAPK1ERBB2
SCHEMBL8316857 0.85 EGFR (0.58) EGFRHTTHIF1ASYKAURKB
SCHEMBL8318926 0.81 EGFR (0.71) EGFRHTTHIF1AMAPK1ERBB2
SCHEMBL8316531 0.80 EGFR (0.68) EGFRHTTHIF1A
SCHEMBL8317938 0.79 EGFR (0.73) EGFRHTTHIF1A
SCHEMBL8316963 0.79 EGFR (0.86) EGFRHTTHIF1AMAPK1ERBB2
SCHEMBL8318660 0.79 EGFR (0.61) EGFRHTTHIF1AMAPK1
SCHEMBL8318090 0.79 EGFR (0.77) EGFRHTTHIF1A
SCHEMBL8315552 0.78 EGFR (0.73) EGFRHTTHIF1AMAPK1ERBB2
SCHEMBL8316168 0.78 EGFR (1.00) EGFRHTTHIF1AMAPK1ERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0779888-B1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM BOEHRINGER INGELHEIM PHARMA (DE) 1999-04-28 EP disclosed
EP-0779888-A1 PYRIMIDO [5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1997-06-25 EP disclosed
WO-1996007657-A1 PYRIMIDO[5,4-D]PYRIMIDINES, DRUGS CONTAINING THESE COMPOUNDS, THEIR USE, AND PROCESS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-03-14 WO disclosed