SCHEMBL8320650

SCHEMBL8320650

CC(C)N(CC#N)C(=O)C(N)C(C)(C)C

nearest known ligand 0.65

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 16/20 0.65
DPP8 Q6V1X1 1/20 0.32
DPP9 Q86TI2 1/20 0.32
CYP1A2 P05177 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326636 0.77 DPP4 (1.00) DPP4DPP8DPP9
SCHEMBL8321440 0.77 DPP4 (1.00) DPP4DPP8DPP9
SCHEMBL14899541 0.73 DPP4 (0.55) DPP4DPP8DPP9
SCHEMBL8320687 0.72 DPP4 (1.00) DPP4DPP8DPP9
SCHEMBL27693121 0.71 DPP4 (1.00) DPP4DPP8DPP9
SCHEMBL2757918 0.71 DPP4 (0.39) DPP4CYP1A2MAPK1
SCHEMBL387066 0.71 DPP4 (1.00) DPP4DPP8DPP9
SCHEMBL18410820 0.71 DPP4 (0.46) DPP4CYP1A2MAPK1
SCHEMBL3298428 0.66 DPP4 (0.37) DPP4CYP1A2MAPK1
SCHEMBL4376489 0.65 DPP4 (0.58) DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1553937-B1 GLYCINENITRILE-BASED INHIBITORS OF DIPEPTIDYL PEPTIDASE IV BRISTOL MYERS SQUIBB CO (US) 2010-06-02 EP disclosed
WO-2004037181-A2 GLYCINENITRILE-BASED INHIBITORS OF DIPEPTIDYL PEPTIDASE IV AND METHODS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-05-06 WO disclosed