Gw832467X

Gw832467X

SCHEMBL8320682

Cc1ccc2c(-c3ccnc(Nc4ccc5c(c4)OCCO5)n3)c(-c3ccc(C(F)(F)F)cc3)nn2n1

nearest known ligand 0.84

Full drug profile on Sugi Atlas →

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 20/20 0.84
CDK2 P24941 3/20 0.84
CDK4 P11802 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4486988 0.92 GSK3B (0.89) GSK3BCDK2CDK4
SCHEMBL4477642 0.91 GSK3B (1.00) GSK3BCDK2CDK4
SCHEMBL4492120 0.91 GSK3B (1.00) GSK3BCDK2CDK4
SCHEMBL4475404 0.89 GSK3B (1.00) GSK3BCDK2CDK4
Gw828525X SCHEMBL4472561 0.88 GSK3B (0.85) GSK3BCDK2
SCHEMBL4491810 0.84 GSK3B (0.82) GSK3BCDK2
SCHEMBL4475079 0.80 GSK3B (1.00) GSK3BCDK2CDK4
Gw827102X SCHEMBL4474674 0.80 GSK3B (1.00) GSK3BCDK2CDK4
Gw829906X SCHEMBL4476648 0.80 GSK3B (1.00) GSK3BCDK2CDK4
SCHEMBL4474335 0.79 GSK3B (0.91) GSK3BCDK2CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582630-B2 Pyradazine compounds as GSK-3 inhibitors SMITHKLINE BEECHAM CORPORATION (US) 2009-09-01 US disclosed
WO-2004035588-A1 PYRADAZINE COMPOUNDS AS GSK-3 INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2004-04-29 WO disclosed