SCHEMBL8324857

SCHEMBL8324857

CC1CCN(C(=O)c2cc3ncnc(NC(C)c4nc5cc(Cl)ccc5[nH]4)c3cc2Cl)C1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EGFR P00533 6/20 0.37
CNR1 P21554 10/20 0.37
ERBB2 P04626 2/20 0.37
CNR2 P34972 6/20 0.36
HPGD P15428 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
GRM5 P41594 1/20 0.35
HRH4 Q9H3N8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4149878 0.95 HPGD (0.39) EGFRCNR1ERBB2CNR2HPGD
SCHEMBL14073985 0.92 PAK4 (0.38) EGFRCNR1ERBB2CNR2
SCHEMBL4163815 0.92 PAK4 (0.38) EGFRCNR1ERBB2CNR2
SCHEMBL4163812 0.92 PAK4 (0.38) EGFRCNR1ERBB2CNR2
SCHEMBL13772343 0.92 PAK4 (0.38) EGFRCNR1ERBB2CNR2
SCHEMBL4148898 0.91 EPHA2 (0.38) EGFR
SCHEMBL4148894 0.91 EPHA2 (0.38) EGFR
SCHEMBL8325093 0.91 EPHA2 (0.38) EGFR
SCHEMBL4150065 0.91 PAK4 (0.40) EGFRCNR1ERBB2CNR2
SCHEMBL6262544 0.90 EGFR (0.40) EGFRCNR1ERBB2CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004058743-A1 NOVEL SUBSTITUTED NITROGEN-CONTAINING HETEROBICYCLES AND USE THEREOF AS FACTOR XA INHIBITORS BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2004-07-15 WO disclosed