SCHEMBL8325614

SCHEMBL8325614

CN[C@H](C)[C@H]1CCN(c2c(F)cc3c(=O)c(OC(=O)O)cn(C4CC4)c3c2OC)C1

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.67
KDM4E B2RXH2 9/20 0.55
HPGD P15428 4/20 0.55
ALDH1A1 P00352 4/20 0.55
HSD17B10 Q99714 2/20 0.55
POLB P06746 2/20 0.55
TDP1 Q9NUW8 2/20 0.55
PRKD3 O94806 1/20 0.55
ALOX15 P16050 1/20 0.55
OPRM1 P35372 1/20 0.55
CLK2 P49760 1/20 0.55
CLK4 Q9HAZ1 1/20 0.55
LMNA P02545 2/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
CYP2C19 P33261 1/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
ATM Q13315 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326332 1.00 KCNH2 (0.67) KCNH2KDM4EHPGDALDH1A1HSD17B10
SCHEMBL8331786 1.00 KCNH2 (0.67) KCNH2KDM4EHPGDALDH1A1HSD17B10
SCHEMBL8329535 0.92 KCNH2 (0.56) KCNH2KDM4EHPGDALDH1A1HSD17B10
SCHEMBL8328878 0.92 KCNH2 (0.65) KCNH2KDM4EHPGDALDH1A1HSD17B10
SCHEMBL8328599 0.92 KCNH2 (0.56) KCNH2KDM4EHPGDALDH1A1HSD17B10
SCHEMBL8329691 0.92 KCNH2 (0.56) KCNH2KDM4EHPGDALDH1A1HSD17B10
SCHEMBL8330117 0.92 KCNH2 (0.65) KCNH2KDM4EHPGDALDH1A1HSD17B10
SCHEMBL9689745 0.92 KCNH2 (0.55) KCNH2KDM4EHPGDALDH1A1HSD17B10
Premafloxacin SCHEMBL8324081 0.90 KCNH2 (0.81) KCNH2KDM4EHPGDALDH1A1HSD17B10
Premafloxacin SCHEMBL7983357 0.90 KCNH2 (0.81) KCNH2KDM4EHPGDALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0559774-B1 INDIVIDUAL STEREOISOMERS OF 7- 3-(1-AMINOALKYL)-1-PYRROLIDINYL]-QUINOLONES AND NAPHTHYRIDONES AS ANTIBACTERIAL AGENTS WARNER LAMBERT CO (US) 1999-07-07 EP claimed