Bromide

Bromide

SCHEMBL8325666

Br.CCN(OCCO)c1nc(-c2ccc(F)c3ccccc23)cc(C(C)C)n1

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR1B known ✓ P28222 1/20 0.53
HTR2B P41595 1/20 0.53
GPR65 Q8IYL9 1/20 0.53
CRHR1 P34998 2/20 0.34
DYRK1A Q13627 1/20 0.32
ALOX5AP P20292 2/20 0.31
FEN1 P39748 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8580284 0.78 HTR1B (0.58) HTR1BHTR2BGPR65CRHR1DYRK1A
SCHEMBL5750446 0.78 HTR1B (0.67) HTR1BHTR2BGPR65CRHR1DYRK1A
Bromide SCHEMBL5750327 0.76 HTR1B (0.53) HTR1BHTR2BGPR65ALOX5APFEN1
Bromide SCHEMBL5750336 0.75 HTR1B (0.52) HTR1BHTR2BGPR65
SCHEMBL5746220 0.73 HTR1B (0.53) HTR1BHTR2BGPR65
Bromide SCHEMBL8386216 0.73 HTR1B (0.58) HTR1BHTR2BGPR65
SCHEMBL5745868 0.73 HTR1B (0.58) HTR1BHTR2BGPR65DYRK1A
SCHEMBL5749062 0.73 HTR1B (0.60) HTR1BHTR2BGPR65CRHR1DYRK1A
Hydrochloric Acid SCHEMBL5750473 0.71 HTR1B (0.58) HTR1BHTR2BGPR65
SCHEMBL5747074 0.71 HTR1B (0.58) HTR1BHTR2BGPR65DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901474-A1 ARYL PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-03-17 EP disclosed
WO-1997044326-A1 ARYL PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-11-27 WO disclosed