SCHEMBL8328730

SCHEMBL8328730

CN(C)C1CCC(NC(=O)OC(C)(C)C)C1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.55
KDM1A O60341 1/20 0.45
MAOB P27338 1/20 0.45
CTSK P43235 2/20 0.44
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
HSD11B1 P28845 2/20 0.40
CYP2C9 P11712 1/20 0.40
KMT2A Q03164 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GAA P10253 2/20 0.40
DRD2 P14416 2/20 0.40
EPHX1 P07099 1/20 0.39
EPHX2 P34913 1/20 0.39
REN P00797 1/20 0.39
JAK1 P23458 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24335931 1.00 BTK (0.55) BTKKDM1AMAOBCTSKNFKB1
SCHEMBL8611872 1.00 BTK (0.55) BTKKDM1AMAOBCTSKNFKB1
SCHEMBL22200775 0.92 BTK (0.66) BTKKDM1AMAOBCTSKNFKB1
SCHEMBL4590525 0.90 BTK (0.50) BTKKDM1AMAOBCTSKNFKB1
SCHEMBL626875 0.90 BTK (0.50) BTKKDM1AMAOBCTSKNFKB1
SCHEMBL626874 0.90 BTK (0.50) BTKKDM1AMAOBCTSKNFKB1
SCHEMBL28735308 0.88 BTK (0.51) BTKKDM1AMAOBCTSKNFKB1
SCHEMBL28735448 0.88 BTK (0.51) BTKKDM1AMAOBCTSKNFKB1
SCHEMBL22200605 0.83 BTK (0.50) BTKKDM1AMAOBCTSKNFKB1
SCHEMBL28621935 0.83 BTK (0.53) BTKKDM1AMAOBCTSKNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5925624-A ANTIINFLAMMATORY AGENTS TREATING PATIENTS WITH INFLAMMATORY CONDITIONS SUSCEPTIBLE TO LEUKOCYTE-INDUCED TISSUE DAMAGE GLAXO GROUP LIMITED (GB) 1999-07-20 US disclosed
US-5889178-A N-(2,2-DIPHENYLETHYL)-DERIVATIVES GLAXO GROUP LIMITED (GB) 1999-03-30 US disclosed
EP-0680488-B1 2,6-DIAMINOPURINE DERIVATIVES GLAXO GROUP LTD (GB) 1998-04-08 EP disclosed