SCHEMBL8329134

SCHEMBL8329134

CC(C)(C)OC(=O)N(CCN)CCN(Cc1ccc(F)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 2/20 0.46
SSTR4 P31391 1/20 0.42
HDAC3 O15379 2/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC2 Q92769 2/20 0.41
NCOR2 Q9Y618 2/20 0.41
KCNQ4 P56696 3/20 0.41
KCNQ5 Q9NR82 3/20 0.41
RIPK1 Q13546 2/20 0.41
GRM2 Q14416 1/20 0.41
KDM1A O60341 3/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
NR1D1 P20393 1/20 0.39
YAP1 P46937 1/20 0.38
TEAD4 Q15561 1/20 0.38
TEAD2 Q15562 1/20 0.38
POLB P06746 1/20 0.38
APEX1 P27695 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2259362 0.97 ROCK1 (0.48) ROCK1SSTR4HDAC3HDAC1HDAC2
SCHEMBL8329242 0.95 ROCK1 (0.45) ROCK1SSTR4HDAC3HDAC1HDAC2
SCHEMBL8331481 0.90 SSTR4 (0.42) ROCK1SSTR4HDAC3HDAC1HDAC2
SCHEMBL8328955 0.88 HDAC3 (0.43) ROCK1SSTR4HDAC3HDAC1HDAC2
SCHEMBL2257781 0.88 AOC3 (0.43) ROCK1SSTR4KCNQ4KCNQ5GRM2
SCHEMBL8325749 0.88 SSTR4 (0.54) SSTR4HDAC3HDAC1HDAC2NCOR2
SCHEMBL8329746 0.87 SOAT1 (0.43) ROCK1SSTR4HDAC3HDAC1HDAC2
SCHEMBL7497944 0.86 SSTR4 (0.40) ROCK1SSTR4HDAC3HDAC1HDAC2
SCHEMBL4744310 0.85 SSTR4 (0.56) SSTR4HDAC3HDAC1HDAC2NCOR2
SCHEMBL2261679 0.84 HDAC3 (0.44) SSTR4HDAC3HDAC1HDAC2NCOR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
US-5736550-A TREATMENT OF GASTROINTESTINAL TRACT DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-04-07 US disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed