SCHEMBL8333311

SCHEMBL8333311

COc1cc(-n2ccnc2)cc(C(F)(F)F)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 4/20 0.55
CYP11B2 P19099 4/20 0.55
ALDH1A1 P00352 3/20 0.49
TDP1 Q9NUW8 3/20 0.49
KMT2A Q03164 2/20 0.49
KDM4E B2RXH2 1/20 0.49
MAOA P21397 2/20 0.44
MAOB P27338 2/20 0.44
CYP19A1 P11511 5/20 0.43
CYP3A4 P08684 4/20 0.41
CYP1A2 P05177 3/20 0.41
CYP2D6 P10635 3/20 0.41
CYP2C19 P33261 3/20 0.41
CYP2C9 P11712 2/20 0.41
HTT P42858 1/20 0.41
LMNA P02545 3/20 0.41
MAPT P10636 3/20 0.41
MAPK1 P28482 2/20 0.41
MEN1 O00255 1/20 0.41
PMP22 Q01453 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14483736 0.84 CYP11B1 (0.68) CYP11B1CYP11B2TDP1MAOAMAOB
SCHEMBL18290496 0.84 CYP3A4 (0.47) CYP11B1CYP11B2ALDH1A1TDP1KMT2A
SCHEMBL1882019 0.84 CYP3A4 (0.47) CYP11B1CYP11B2ALDH1A1TDP1KMT2A
SCHEMBL31138008 0.84 CYP11B1 (0.68) CYP11B1CYP11B2TDP1MAOAMAOB
Hydrochloric Acid SCHEMBL17583800 0.82 CYP3A4 (0.46) CYP11B1CYP11B2ALDH1A1TDP1KMT2A
SCHEMBL14092962 0.80 CYP3A4 (0.41) CYP11B1CYP11B2ALDH1A1TDP1KMT2A
SCHEMBL10104435 0.80 NR2E1 (0.42) CYP11B1CYP11B2ALDH1A1TDP1KMT2A
Hydrochloric Acid SCHEMBL4425277 0.78 CYP19A1 (0.48) CYP11B1ALDH1A1KMT2ACYP19A1MEN1
SCHEMBL588961 0.77 NR2E1 (0.56) CYP11B1CYP11B2ALDH1A1TDP1KMT2A
SCHEMBL30880594 0.77 CYP11B1 (0.59) CYP11B1CYP11B2TDP1MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999009845-A1 IMIDAZOQUINOXALINE PROTEIN TYROSINE KINASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 1999-03-04 WO claimed