SCHEMBL8337186

SCHEMBL8337186

Cc1cc(I)cc2[nH]c(C(=O)O)c(/C=C3\CCN(c4ccccc4)C3=O)c12

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 1/20 0.41
GPR17 Q13304 3/20 0.34
ACHE P22303 1/20 0.32
MEN1 O00255 1/20 0.31
LMNA P02545 1/20 0.31
CYP1A2 P05177 1/20 0.31
MAPK1 P28482 1/20 0.31
BLM P54132 1/20 0.31
PMP22 Q01453 1/20 0.31
KMT2A Q03164 1/20 0.31
PPARG P37231 1/20 0.31
PPARD Q03181 1/20 0.31
PPARA Q07869 1/20 0.31
NPC1 O15118 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL499308 0.81 GRIN1 (0.59) GRIN1GPR17MEN1LMNACYP1A2
SCHEMBL499309 0.81 GRIN1 (0.59) GRIN1GPR17MEN1LMNACYP1A2
SCHEMBL4422661 0.80 GRIN1 (0.58) GRIN1GPR17MEN1LMNACYP1A2
SCHEMBL4422653 0.80 GRIN1 (0.58) GRIN1GPR17MEN1LMNACYP1A2
SCHEMBL8190768 0.76 GRIN1 (0.55) GRIN1GPR17MEN1LMNACYP1A2
SCHEMBL8190756 0.76 GRIN1 (0.55) GRIN1GPR17MEN1LMNACYP1A2
SCHEMBL8181067 0.75 GRIN1 (0.54) GRIN1GPR17MEN1LMNACYP1A2
SCHEMBL8181079 0.75 GRIN1 (0.54) GRIN1GPR17MEN1LMNACYP1A2
SCHEMBL1720270 0.73 GRIN1 (0.52) GRIN1MEN1LMNACYP1A2MAPK1
SCHEMBL30521938 0.73 GRIN1 (0.52) GRIN1MEN1LMNACYP1A2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004039371-A2 COMPOSITIONS OF CYCLOOXYGENASE-2 SELECTIVE INHIBITORS AND NMDA RECEPTOR ANTAGONISTS FOR THE TREATMENT OR PREVENTION OF NEUROPATHIC PAIN PHARMACIA CORPORATION (US) 2004-05-13 WO disclosed