SCHEMBL8344854

SCHEMBL8344854

CN(C)c1ccc(NC2CCN(c3nc(-c4ccncn4)cc(=O)n3C)CC2)cc1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 20/20 0.61
CYP2D6 P10635 5/20 0.49
CYP1A2 P05177 3/20 0.47
CSNK1A1 P48729 1/20 0.47
GSK3A P49840 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13915154 0.87 GSK3B (0.48) GSK3BCYP2D6CYP1A2
SCHEMBL13917298 0.87 GSK3B (0.61) GSK3BCYP2D6CYP1A2
SCHEMBL698301 0.84 GSK3B (0.64) GSK3BCYP2D6CYP1A2CSNK1A1GSK3A
SCHEMBL696475 0.84 GSK3B (0.64) GSK3BCYP2D6CYP1A2CSNK1A1GSK3A
SCHEMBL13711419 0.83 GSK3B (0.62) GSK3BCYP2D6CYP1A2
SCHEMBL697014 0.83 GSK3B (0.62) GSK3BCYP2D6CYP1A2
SCHEMBL87819 0.83 GSK3B (0.51) GSK3BCYP2D6CYP1A2
SCHEMBL8234787 0.82 GSK3B (0.65) GSK3BCYP2D6CYP1A2
SCHEMBL697865 0.82 GSK3B (0.65) GSK3BCYP2D6CYP1A2
SCHEMBL13917296 0.81 GSK3B (0.61) GSK3BCYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504411-B2 2,3,6-Trisubstituted-4-pyrimidone derivatives MITSUBISHI TANABE PHARMA CORPORATION (JP) 2009-03-17 US disclosed
US-7504411-B2 2,3,6-Trisubstituted-4-pyrimidone derivatives MITSUBISHI TANABE PHARMA CORPORATION (JP) 2009-03-17 US disclosed
WO-2004085408-A1 2, 3, 6-TRISUBSTITUTED-4-PYRIMIDONE DERIVATIVES MITSUBISHI PHARMA CORPORATION (JP) 2004-10-07 WO disclosed