SCHEMBL8345170

SCHEMBL8345170

CCOC(=O)CC(=O)NCCN1CCOCC1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.55
POLB P06746 2/20 0.54
TDP1 Q9NUW8 1/20 0.54
CYP3A4 P08684 1/20 0.52
LMNA P02545 1/20 0.51
HSD17B10 Q99714 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.49
MAPK1 P28482 1/20 0.48
HBB P68871 1/20 0.48
KMT2A Q03164 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2759481 0.83 TDP1 (0.57) TSHRPOLBTDP1CYP3A4
SCHEMBL2039034 0.83 TDP1 (0.51) TSHRPOLBTDP1CYP3A4LMNA
SCHEMBL84933 0.81 TSHR (0.59) TSHRPOLBTDP1HSD17B10SMN1; SMN2
SCHEMBL3470544 0.81 TDP1 (0.62) TSHRPOLBTDP1CYP3A4LMNA
SCHEMBL12465711 0.81 TDP1 (0.48) TSHRPOLBTDP1CYP3A4LMNA
SCHEMBL9602488 0.80 TSHR (0.58) TSHRPOLBTDP1HSD17B10SMN1; SMN2
SCHEMBL85431 0.78 TSHR (0.60) TSHRPOLBTDP1HSD17B10SMN1; SMN2
SCHEMBL65336 0.78 TSHR (0.63) TSHRPOLBTDP1LMNASMN1; SMN2
SCHEMBL28191332 0.78 TSHR (0.56) TSHRPOLBTDP1LMNAHSD17B10
Hydrochloric Acid SCHEMBL5843426 0.77 TSHR (0.62) TSHRPOLBTDP1HSD17B10SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7230017-B2 Dihydropyridinone derivatives BAYER HEALTHCARE AG (DE) 2007-06-12 US disclosed
US-7230017-B2 Dihydropyridinone derivatives BAYER HEALTHCARE AG (DE) 2007-06-12 US disclosed
WO-2004020410-A2 DIHYDROPYRIDINONE DERIVATIVES AS HNE INHIBITORS BAYER HEALTHCARE AG (DE) 2004-03-11 WO disclosed