SCHEMBL8345512

SCHEMBL8345512

CSc1ccc2c(c1)S(=O)(=O)NC2=O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 16/20 0.57
CA9 Q16790 16/20 0.57
CA2 P00918 14/20 0.51
CA7 P43166 8/20 0.51
CA1 P00915 6/20 0.51
GLO1 Q04760 1/20 0.51
KDM4E B2RXH2 1/20 0.50
USP2 O75604 1/20 0.50
LMNA P02545 1/20 0.50
BCHE P06276 1/20 0.50
CA4 P22748 1/20 0.50
CA6 P23280 1/20 0.50
CA5A P35218 1/20 0.50
KMT2A Q03164 1/20 0.50
CA14 Q9ULX7 1/20 0.50
CA5B Q9Y2D0 1/20 0.50
CHEK1 O14757 1/20 0.49
DAPK3 O43293 1/20 0.49
MAP4K4 O95819 1/20 0.49
RET P07949 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7303822 0.79 CA12 (0.53) CA12CA9CA2CA7CA1
SCHEMBL29349483 0.77 CA12 (0.62) CA12CA9CA2CA7CA1
SCHEMBL1249735 0.77 CA12 (0.62) CA12CA9CA2CA7CA1
SCHEMBL29350588 0.73 CA12 (0.62) CA12CA9CA2CA7CA1
SCHEMBL30834838 0.73 CA12 (0.62) CA12CA9CA2CA7CA1
SCHEMBL10815413 0.73 CA12 (0.62) CA12CA9CA2CA7CA1
SCHEMBL6753007 0.73 CHEK1 (0.79) CA12CA9CA2CA7CA1
SCHEMBL1290860 0.73 CA12 (1.00) CA12CA9CA2CA7CA1
SCHEMBL31168119 0.73 CHEK1 (0.79) CA12CA9CA2CA7CA1
SCHEMBL9814710 0.73 CA12 (0.62) CA12CA9CA2CA7CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5856349-A 2-Saccharinylmethyl heterocyclic carboxylates useful as proteolytic enzyme inhibitors and compositions and method of use thereof SANOFI (FR) 1999-01-05 US disclosed