SCHEMBL8348776

SCHEMBL8348776

COc1ccc2c(O[C@@H]3C[C@@H](C(=O)NC4(C(=O)NS(=O)(=O)c5cccs5)CC45CCC5)N(C(=O)[C@@H](NC(=O)OC(C)(C)C)C(C)(C)C)C3)cc(-c3ccccc3)nc2c1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.47
CTSB P07858 2/20 0.39
PPP3CB P16298 1/20 0.39
ELANE P08246 4/20 0.35
ABCC1 P33527 1/20 0.35
ABCC2 Q92887 1/20 0.35
ABCG2 Q9UNQ0 1/20 0.35
USP2 O75604 1/20 0.34
USP8 P40818 1/20 0.34
MCL1 Q07820 1/20 0.34
BIRC2 Q13490 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8349695 0.99 CYP3A4 (0.47) CYP3A4CTSBPPP3CBELANEABCC1
SCHEMBL8348948 0.98 CYP3A4 (0.48) CYP3A4CTSBPPP3CBELANEABCC1
SCHEMBL8349697 0.95 CYP3A4 (0.48) CYP3A4CTSBPPP3CBELANEABCC1
SCHEMBL8348770 0.94 CYP3A4 (0.48) CYP3A4CTSBPPP3CBELANEABCC1
SCHEMBL5693284 0.90 CYP3A4 (0.57) CYP3A4CTSB
SCHEMBL5692578 0.90 CYP3A4 (0.46) CYP3A4CTSBPPP3CBELANEABCC1
SCHEMBL5692629 0.89 CYP3A4 (0.46) CYP3A4CTSBPPP3CBELANEABCC1
SCHEMBL6308074 0.89 CYP3A4 (0.57) CYP3A4CTSB
SCHEMBL2345253 0.89 CYP3A4 (0.62) CYP3A4CTSBPPP3CB
SCHEMBL5692632 0.88 CYP3A4 (0.58) CYP3A4CTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1506000-B9 HETEROCYCLICSULFONAMIDE HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2011-08-31 EP disclosed
EP-1506000-B1 HETEROCYCLICSULFONAMIDE HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2010-09-15 EP disclosed
WO-2003099316-A1 HETEROCYCLICSULFONAMIDE HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-12-04 WO disclosed