SCHEMBL8348951

SCHEMBL8348951

CC(=O)N(Cc1ccccc1O)C1CCC(NC(=O)c2cc(F)cnc2Oc2ccc(F)cc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 17/20 0.53
PDE4A P27815 1/20 0.53
PDE4D Q08499 1/20 0.53
PTGER4 P35408 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6063308 1.00 PDE4B (0.53) PDE4BPDE4APDE4DPTGER4
SCHEMBL8354209 0.91 PDE4B (0.47) PDE4BPDE4APDE4DPTGER4
SCHEMBL8353637 0.87 PDE4B (0.52) PDE4BPDE4APDE4DPTGER4
SCHEMBL6063994 0.87 PDE4B (0.52) PDE4BPDE4APDE4DPTGER4
SCHEMBL6063105 0.86 PDE4B (0.51) PDE4BPDE4APDE4DPTGER4
SCHEMBL8351723 0.86 PDE4B (0.51) PDE4BPDE4APDE4DPTGER4
SCHEMBL6063506 0.84 PDE4B (0.56) PDE4BPDE4APDE4DPTGER4
SCHEMBL8354177 0.84 PDE4B (0.56) PDE4BPDE4APDE4DPTGER4
SCHEMBL6063595 0.82 PDE4B (0.54) PDE4BPDE4APDE4DPTGER4
SCHEMBL8351099 0.82 PDE4B (0.54) PDE4BPDE4APDE4DPTGER4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003068233-A1 NICOTINAMIDE DERIVATIVES AND A TIOTROPIUM SALT IN COMBINATION FOR THE TREATMENT OF E.G. INFLAMMATORY, ALLERGIC AND RESPIRATORY DISEASES PFIZER LIMITED (GB) 2003-08-21 WO disclosed
WO-2003068235-A1 NICOTINAMIDE DERIVATIVES USEFUL AS PDE4 INHIBITORS PFIZER LIMITED (GB) 2003-08-21 WO disclosed