SCHEMBL8349396

SCHEMBL8349396

COC(=O)[C@H]1CC[C@H](NC(=O)c2cc(F)cnc2Oc2ccc(F)cc2)CC1

nearest known ligand 0.59

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 13/20 0.59
PDE4A P27815 1/20 0.59
PDE4D Q08499 1/20 0.59
PTGER4 P35408 5/20 0.50
CNR2 P34972 2/20 0.45
ABHD6 Q9BV23 1/20 0.45
CNR1 P21554 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6062652 1.00 PDE4B (0.59) PDE4BPDE4APDE4DPTGER4CNR2
SCHEMBL6063356 0.89 PDE4B (0.59) PDE4BPDE4APDE4DPTGER4CNR2
SCHEMBL8352461 0.89 PDE4B (0.59) PDE4BPDE4APDE4DPTGER4CNR2
SCHEMBL8352911 0.86 PDE4B (0.60) PDE4BPDE4APDE4DPTGER4CNR2
SCHEMBL6063667 0.86 PDE4B (0.60) PDE4BPDE4APDE4DPTGER4
SCHEMBL8351599 0.86 PDE4B (0.60) PDE4BPDE4APDE4DPTGER4
SCHEMBL6063497 0.86 PDE4B (0.58) PDE4BPDE4APDE4DPTGER4CNR2
SCHEMBL8353587 0.86 PDE4B (0.58) PDE4BPDE4APDE4DPTGER4CNR2
SCHEMBL8353040 0.86 PDE4B (0.58) PDE4BPDE4APDE4DPTGER4CNR2
SCHEMBL6063391 0.86 PDE4B (0.58) PDE4BPDE4APDE4DPTGER4CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003068233-A1 NICOTINAMIDE DERIVATIVES AND A TIOTROPIUM SALT IN COMBINATION FOR THE TREATMENT OF E.G. INFLAMMATORY, ALLERGIC AND RESPIRATORY DISEASES PFIZER LIMITED (GB) 2003-08-21 WO disclosed
WO-2003068235-A1 NICOTINAMIDE DERIVATIVES USEFUL AS PDE4 INHIBITORS PFIZER LIMITED (GB) 2003-08-21 WO disclosed