SCHEMBL835647

SCHEMBL835647

CS(=O)(=O)Nc1cccc(-c2cnn3c(-c4ccnc(-c5ccoc5)c4)cnc3c2)c1

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
FYN P06241 15/20 0.52
KLK7 P49862 1/20 0.45
FGFR1 P11362 1/20 0.41
FGFR3 P22607 1/20 0.41
FLT3 P36888 1/20 0.40
HTT P42858 1/20 0.39
MET P08581 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL836511 0.85 FYN (0.55) FYNKLK7FGFR1FGFR3
SCHEMBL3026322 0.84 FYN (0.54) FYN
SCHEMBL837011 0.83 FYN (0.54) FYNKLK7FGFR1FGFR3HTT
SCHEMBL836186 0.81 FGFR1 (0.65) FYNFGFR1FGFR3FLT3
SCHEMBL835970 0.81 FYN (0.48) FYNFGFR1FGFR3FLT3
SCHEMBL835806 0.81 FYN (0.47) FYN
SCHEMBL834234 0.79 FYN (0.67) FYN
SCHEMBL836996 0.78 FYN (0.58) FYNFGFR1FGFR3
SCHEMBL836699 0.77 FYN (0.53) FYNFGFR1FGFR3
SCHEMBL835261 0.76 FYN (0.48) FYNFGFR1FGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143253-B2 Organic compounds NOVARTIS AG (CH) 2012-03-27 US claimed
EP-2183027-B1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2011-08-31 EP claimed
US-20100204235-A1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2010-08-12 US claimed
EP-2183027-A1 ORGANIC COMPOUNDS Novartis Ag (CH) 2010-05-12 EP claimed
WO-2009013335-A1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2009-01-29 WO claimed
US-8143253-B2 Organic compounds NOVARTIS AG (CH) 2012-03-27 US disclosed
EP-2183027-B1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2011-08-31 EP disclosed
US-20100204235-A1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2010-08-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100204235-A1 ORGANIC COMPOUNDS ALK, OR10J3, FFAR4 FYN 971/4885KLK7 4346/4885FGFR1 20/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.