SCHEMBL8358666

SCHEMBL8358666

COc1cc(C(=O)Nc2nc3c(C)ccc(N4CCOCC4)c3s2)ccn1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 18/20 0.51
ADORA1 P30542 12/20 0.51
ADORA2B P29275 4/20 0.51
ADORA3 P0DMS8 2/20 0.51
MAPT P10636 2/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C19 P33261 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5560780 0.91 ADORA2A (0.63) ADORA2AADORA1ADORA2BADORA3
SCHEMBL5561440 0.84 ADORA2A (0.59) ADORA2AADORA1ADORA2BADORA3
SCHEMBL3048203 0.84 ADORA2A (0.63) ADORA2AADORA1ADORA2BADORA3
SCHEMBL5560995 0.84 ADORA2A (0.59) ADORA2AADORA1ADORA2BADORA3
SCHEMBL5561019 0.84 ADORA2A (0.63) ADORA2AADORA1ADORA2BADORA3
SCHEMBL5566040 0.83 ADORA2A (0.62) ADORA2AADORA1ADORA2BADORA3
SCHEMBL5566933 0.83 ADORA2A (0.58) ADORA2AADORA1ADORA2BADORA3
SCHEMBL5558477 0.82 ADORA2A (0.75) ADORA2AADORA1ADORA2BADORA3MAPT
SCHEMBL5561416 0.82 ADORA2A (0.58) ADORA2AADORA1ADORA2BADORA3
SCHEMBL5561585 0.82 ADORA2A (0.56) ADORA2AADORA1ADORA2BADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003043634-A1 BENZOTHIAZOLE DERIVATIVES AS ADENOSINE RECEPTOR LIGANDS F. HOFFMANN-LA ROCHE AG (CH) 2003-05-30 WO disclosed