SCHEMBL8359571

SCHEMBL8359571

N#Cc1ccccc1Cn1cncc1CC(N)=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.46
ALDH1A1 P00352 5/20 0.44
GALR3 O60755 1/20 0.44
RAB9A P51151 1/20 0.44
TSHR P16473 4/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
MAPT P10636 3/20 0.42
SIRT2 Q8IXJ6 1/20 0.41
SIRT1 Q96EB6 1/20 0.41
LMNA P02545 1/20 0.41
CYP11B1 P15538 3/20 0.40
CYP11B2 P19099 3/20 0.40
NPSR1 Q6W5P4 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
HPGD P15428 1/20 0.39
KMT2A Q03164 1/20 0.39
GAA P10253 1/20 0.39
HSD17B10 Q99714 1/20 0.39
FNTA P49354 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12820668 0.83 CYP11B1 (0.58) CYP19A1ALDH1A1GALR3RAB9ATSHR
SCHEMBL8441652 0.81 CYP19A1 (0.49) CYP19A1ALDH1A1GALR3RAB9ATSHR
SCHEMBL9267101 0.77 CYP11B1 (0.58) ALDH1A1TSHRCYP11B1CYP11B2GAA
SCHEMBL7478451 0.77 CYP11B1 (0.69) CYP19A1CYP11B1CYP11B2FNTAFNTB
Hydrochloric Acid SCHEMBL7802265 0.76 CYP11B1 (0.67) CYP19A1CYP11B1CYP11B2FNTAFNTB
Hydrochloric Acid SCHEMBL7473105 0.76 CYP11B1 (0.67) CYP19A1CYP11B1CYP11B2FNTAFNTB
Hydrochloric Acid SCHEMBL7847528 0.76 CYP19A1 (0.52) CYP19A1ALDH1A1GALR3RAB9ATSHR
SCHEMBL27855265 0.75 CYP11B1 (0.48) CYP19A1ALDH1A1GALR3RAB9ASMN1; SMN2
SCHEMBL1064583 0.74 SIRT2 (0.45) CYP19A1ALDH1A1GALR3RAB9ATSHR
SCHEMBL1950222 0.72 CYP11B1 (0.63) CYP19A1ALDH1A1GALR3RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5874452-A Biheteroaryl inhibitors of farnesyl-protein transferase MERCK & CO., INC. (US) 1999-02-23 US disclosed
US-5859035-A Arylheteroaryl inhibitors of farnesyl-protein transferase MERCK & CO., INC. (US) 1999-01-12 US disclosed
US-5854265-A Biheteroaryl inhibitors of farnesyl-protein transferase MERCK & CO., INC. (US) 1998-12-29 US disclosed