SCHEMBL8359596

SCHEMBL8359596

O=C(CCCN1CC=CCC1)N1CCc2[nH]c(=O)c3ccccc3c2C1

nearest known ligand 0.75

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 13/20 0.75
TAAR1 Q96RJ0 1/20 0.53
MAPT P10636 2/20 0.43
GAA P10253 1/20 0.43
ALDH1A1 P00352 2/20 0.42
CASP1 P29466 2/20 0.42
CASP7 P55210 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.41
ALOX15 P16050 1/20 0.41
KMT2A Q03164 1/20 0.41
LMNA P02545 1/20 0.41
BAZ2B Q9UIF8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8362904 0.94 PARP1 (0.74) PARP1TAAR1MAPTGAAALDH1A1
SCHEMBL8363084 0.88 PARP1 (0.73) PARP1TAAR1MAPTGAAALDH1A1
SCHEMBL8359714 0.86 PARP1 (0.84) PARP1TAAR1MAPTGAAALDH1A1
SCHEMBL8359463 0.86 PARP1 (1.00) PARP1TAAR1ALDH1A1KDM4E
SCHEMBL8362893 0.85 PARP1 (0.83) PARP1TAAR1MAPTGAAALDH1A1
SCHEMBL8362897 0.85 PARP1 (0.83) PARP1TAAR1MAPTGAAALDH1A1
SCHEMBL14444067 0.81 PARP1 (0.73) PARP1TAAR1MAPTALDH1A1CASP1
SCHEMBL8359597 0.80 PARP1 (0.74) PARP1TAAR1MAPTGAAALDH1A1
SCHEMBL14444062 0.80 PARP1 (0.73) PARP1TAAR1MAPTGAAALDH1A1
SCHEMBL8363088 0.80 PARP1 (0.73) PARP1MAPTGAAALDH1A1CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003014121-A9 COMPOUNDS, DERIVATIVES, COMPOSITIONS, PREPARATION AND USES GUILFORD PHARM INC (US) 2004-03-25 WO disclosed
WO-2003014121-A1 COMPOUNDS, DERIVATIVES, COMPOSITIONS, PREPARATION AND USES GUILFORD PHARMACEUTICALS INC. (US) 2003-02-20 WO disclosed