SCHEMBL8359797

SCHEMBL8359797

CCOc1ccc(-n2c(C)c3c(C)nnc(CCC(=O)O)c3c2C)cc1

nearest known ligand 0.72

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 20/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8359787 0.94 CACNA2D1 (0.74) CACNA2D1
SCHEMBL5009827 0.93 CACNA2D1 (0.72) CACNA2D1
SCHEMBL8360423 0.89 CACNA2D1 (0.69) CACNA2D1
SCHEMBL8359788 0.87 CACNA2D1 (0.66) CACNA2D1
SCHEMBL5008062 0.86 CACNA2D1 (0.71) CACNA2D1
Potassium Ion SCHEMBL5009829 0.86 CACNA2D1 (0.71) CACNA2D1
SCHEMBL5005069 0.84 CACNA2D1 (0.69) CACNA2D1
SCHEMBL5004664 0.84 CACNA2D1 (1.00) CACNA2D1
SCHEMBL6194723 0.84 CACNA2D1 (0.72) CACNA2D1
SCHEMBL5004885 0.83 CACNA2D1 (1.00) CACNA2D1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7465730-B2 Treatment of neuropathic pain with 6H-pyrrolo[3,4-d]pyridazine compounds MERCK & CO. INC. (US) 2008-12-16 US disclosed
US-7465730-B2 Treatment of neuropathic pain with 6H-pyrrolo[3,4-d]pyridazine compounds MERCK & CO. INC. (US) 2008-12-16 US disclosed
WO-2004006836-A2 TREATMENT OF NEUROPATHIC PAIN WITH 6H-PYRROLO[3,4-D]PYRIDAZINE COMPOUNDS MERCK & CO., INC. (US) 2004-01-22 WO disclosed