SCHEMBL8360443

SCHEMBL8360443

CC(C)c1cc(-c2cccc(CC(c3ccccc3)c3ccc([S+](C)[O-])cc3)c2)c2ncccc2c1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 19/20 0.61
PDE4B Q07343 19/20 0.61
PDE4C Q08493 19/20 0.61
PDE4D Q08499 19/20 0.61
CYP2C9 P11712 11/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8343973 0.85 PDE4A (0.61) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL6604913 0.81 PDE4A (0.84) PDE4APDE4BPDE4CPDE4DCYP2C9
Bromide SCHEMBL4031335 0.77 PDE4A (0.59) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL6180752 0.76 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL4025781 0.76 PDE4A (0.66) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL4027089 0.76 PDE4A (0.62) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL4037954 0.76 PDE4A (0.57) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL5257490 0.76 PDE4A (0.57) PDE4APDE4BPDE4CPDE4DCYP2C9
SCHEMBL7448426 0.75 PDE4A (0.56) PDE4APDE4BPDE4CPDE4D
SCHEMBL6184825 0.75 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003105815-A1 COMBINATION OF PDE-V INHIBITORS AND NK1 ANTAGONISTS FOR THE TREATMENT OF DEPRESSION PFIZER PRODUCTS INC. (US) 2003-12-24 WO disclosed