SCHEMBL8364417

SCHEMBL8364417

CS(=O)(=O)CCNCCCc1ccc2c(Nc3ccc(OCc4ccccc4)cc3)ncnc2c1

nearest known ligand 0.74

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
EGFR P00533 16/20 0.74
ERBB2 P04626 15/20 0.74
CHEK2 O96017 1/20 0.56
ROS1 P08922 1/20 0.56
FLT3 P36888 1/20 0.56
ERBB4 Q15303 1/20 0.56
AURKB Q96GD4 1/20 0.56
CLK4 Q9HAZ1 1/20 0.56
MKNK2 Q9HBH9 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8363336 0.97 EGFR (0.75) EGFRERBB2CHEK2ROS1FLT3
SCHEMBL8367286 0.95 EGFR (0.71) EGFRERBB2CHEK2ROS1FLT3
SCHEMBL8367607 0.93 EGFR (0.82) EGFRERBB2
SCHEMBL8364155 0.91 EGFR (0.83) EGFRERBB2
SCHEMBL8368189 0.90 EGFR (0.87) EGFRERBB2CHEK2ROS1FLT3
SCHEMBL8367097 0.90 EGFR (0.76) EGFRERBB2CHEK2ROS1FLT3
SCHEMBL8361665 0.90 EGFR (0.87) EGFRERBB2CHEK2ROS1FLT3
SCHEMBL8361544 0.90 EGFR (0.74) EGFRERBB2CHEK2ROS1FLT3
SCHEMBL8367614 0.88 EGFR (0.79) EGFRERBB2CHEK2ROS1FLT3
SCHEMBL8367271 0.88 EGFR (0.82) EGFRERBB2CHEK2ROS1FLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999035132-A1 HETEROCYCLIC COMPOUNDS GLAXO GROUP LIMITED (GB) 1999-07-15 WO disclosed