SCHEMBL8364786

SCHEMBL8364786

CCCN(CCC)C(=O)c1cc(C)cc(C(=O)N[C@@H](Cc2cc(F)cc(F)c2)[C@@H](O)CS)c1

nearest known ligand 0.71

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.71
BACE2 Q9Y5Z0 6/20 0.71
CTSD P07339 2/20 0.68
CTSE P14091 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5363946 0.92 BACE1 (0.74) BACE1BACE2CTSDCTSE
SCHEMBL4891462 0.90 BACE1 (0.71) BACE1BACE2CTSD
SCHEMBL3351740 0.90 BACE1 (0.71) BACE1BACE2CTSD
SCHEMBL4899242 0.89 BACE1 (0.76) BACE1BACE2CTSD
SCHEMBL5180653 0.89 BACE1 (0.76) BACE1BACE2CTSD
SCHEMBL5579146 0.88 BACE1 (0.69) BACE1BACE2CTSD
SCHEMBL3350491 0.88 BACE1 (0.77) BACE1BACE2CTSDCTSE
SCHEMBL3354515 0.88 BACE1 (0.80) BACE1BACE2CTSD
SCHEMBL3350500 0.88 BACE1 (0.77) BACE1BACE2CTSDCTSE
SCHEMBL5367552 0.88 BACE1 (0.69) BACE1BACE2CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003002122-A1 BETA-HYDROXYAMINE DERIVATIVES USEFUL IN TREATMENT OF ALZHEIMER'S DISEASE ELAN PHARMACEUTICALS, INC. (US) 2003-01-09 WO disclosed