SCHEMBL8364974

SCHEMBL8364974

CCCN(CCC)C(=O)c1cc(C)cc(C(=O)N[C@@H](Cc2cc(F)cc(F)c2)C(O)CCc2ccccc2)c1

nearest known ligand 0.78

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.78
BACE2 Q9Y5Z0 10/20 0.78
CTSD P07339 6/20 0.70
CTSE P14091 4/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3351671 0.91 BACE1 (0.78) BACE1BACE2CTSD
SCHEMBL5374257 0.90 BACE1 (0.69) BACE1BACE2CTSDCTSE
SCHEMBL3351088 0.90 BACE1 (0.84) BACE1BACE2CTSDCTSE
SCHEMBL5380451 0.90 BACE1 (0.69) BACE1BACE2CTSDCTSE
SCHEMBL3354946 0.90 BACE1 (0.73) BACE1BACE2CTSDCTSE
SCHEMBL14541333 0.90 BACE1 (0.73) BACE1BACE2CTSDCTSE
SCHEMBL3353553 0.89 BACE1 (0.83) BACE1BACE2CTSD
SCHEMBL5377987 0.88 BACE1 (0.82) BACE1BACE2CTSD
SCHEMBL5372988 0.88 BACE1 (0.71) BACE1BACE2CTSDCTSE
SCHEMBL6044289 0.88 BACE1 (0.66) BACE1BACE2CTSDCTSE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003002122-A1 BETA-HYDROXYAMINE DERIVATIVES USEFUL IN TREATMENT OF ALZHEIMER'S DISEASE ELAN PHARMACEUTICALS, INC. (US) 2003-01-09 WO disclosed