Ethylene

Ethylene

SCHEMBL8378170

C=C.CCNC(=O)N1CCC(=O)CC1

nearest known ligand 0.64

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.64
HTT P42858 2/20 0.55
FAAH O00519 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
TSHR P16473 1/20 0.41
ALOX12 P18054 1/20 0.41
MAPK1 P28482 1/20 0.41
MTOR P42345 1/20 0.41
RAB9A P51151 1/20 0.41
MEN1 O00255 1/20 0.40
BLM P54132 1/20 0.40
PMP22 Q01453 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
BRD4 O60885 1/20 0.39
PKM P14618 1/20 0.38
MTNR1B P49286 3/20 0.38
MTNR1A P48039 1/20 0.38
POLB P06746 1/20 0.37
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4345849 0.96 KMT2A (0.69) KMT2AHTTFAAHCYP3A4CYP2D6
SCHEMBL10808716 0.81 KMT2A (0.53) KMT2AHTTMAPK1MEN1POLB
SCHEMBL2948216 0.76 KMT2A (0.62) KMT2AHTTFAAHCYP3A4CYP2D6
SCHEMBL4534029 0.76 KMT2A (0.83) KMT2AHTTFAAHCYP3A4CYP2D6
SCHEMBL965286 0.76 KMT2A (0.82) KMT2AHTTMAPK1RAB9APOLB
SCHEMBL19741751 0.76
SCHEMBL17273858 0.74 KMT2A (0.78) KMT2AHTTMAPK1RAB9AMEN1
SCHEMBL4803949 0.74 KMT2A (0.78) KMT2AHTTMAPK1RAB9AMEN1
SCHEMBL966438 0.74 KMT2A (0.78) KMT2AHTTMAPK1RAB9AMEN1
SCHEMBL13674468 0.72 KMT2A (0.83) KMT2AHTTFAAHCYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5883102-A Pharmaceutically active compounds ASTRA PHARMACEUTICALS LIMITED (GB) 1999-03-16 US disclosed
EP-0858451-A1 PHARMACEUTICALLY ACTIVE QUINAZOLINE COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-08-19 EP disclosed
WO-1997014686-A1 PHARMACEUTICALLY ACTIVE QUINAZOLINE COMPOUNDS ASTRA PHARMACEUTICALS LIMITED (GB) 1997-04-24 WO disclosed