SCHEMBL8380917

SCHEMBL8380917

CCSc1nc(N)c(Cc2ccccc2OC)c(N)n1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 7/20 0.54
HTR2C P28335 7/20 0.54
PNP P00491 1/20 0.44
LTA4H P09960 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
TLR7 Q9NYK1 1/20 0.42
ABCB1 P08183 1/20 0.41
IDO1 P14902 2/20 0.41
TAAR1 Q96RJ0 1/20 0.41
ADORA2A P29274 2/20 0.40
ADORA1 P30542 2/20 0.40
ADORA3 P0DMS8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8378051 0.80 HTR2A (0.59) HTR2AHTR2CSMN1; SMN2ADORA2AADORA1
SCHEMBL7096925 0.80 PNP (0.48) HTR2AHTR2CPNPLTA4HTLR7
Hydrochloric Acid SCHEMBL8380954 0.79 HTR2A (0.58) HTR2AHTR2CSMN1; SMN2ADORA2AADORA1
SCHEMBL7094111 0.78 PNP (0.47) HTR2AHTR2CPNPLTA4HTLR7
SCHEMBL7099072 0.77 HTR2A (0.69) HTR2AHTR2C
Hydrochloric Acid SCHEMBL7097008 0.76 HTR2A (0.65) HTR2AHTR2C
SCHEMBL8379832 0.76 ADORA2A (0.50) HTR2AHTR2CSMN1; SMN2ABCB1ADORA2A
Hydrochloric Acid SCHEMBL7095911 0.75 HTR2A (0.52) HTR2AHTR2C
Hydrochloric Acid SCHEMBL7093513 0.75 HTR2A (0.61) HTR2AHTR2C
Hydrochloric Acid SCHEMBL7093698 0.75 HTR2A (0.63) HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901473-A1 NOVEL PIPERAZINYLALKYLTHIOPYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AND A PROCESS FOR THE PREPARATION OF THE NOVEL COMPOUNDS EGIS GYOGYSZERGYAR RT. (HU) 1999-03-17 EP disclosed
WO-1997016429-A1 NOVEL PIPERAZINYLALKYLTHIOPYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AND A PROCESS FOR THE PREPARATION OF THE NOVEL COMPOUNDS EGIS Gyógyszergyár Rt. (HU) 1997-05-09 WO disclosed