SCHEMBL8386147

SCHEMBL8386147

N#C/[C]=[C]/c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.52
APP P05067 1/20 0.43
MAOB P27338 2/20 0.34
MAOA P21397 1/20 0.34
MAPT P10636 3/20 0.33
CYP1A2 P05177 3/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32
THPO P40225 1/20 0.32
TRPA1 O75762 1/20 0.32
ALDH1A1 P00352 4/20 0.31
BLM P54132 1/20 0.31
PMP22 Q01453 1/20 0.31
GRM5 P41594 1/20 0.31
CYP1A1 P04798 1/20 0.31
CYP1B1 Q16678 1/20 0.31
KDM4E B2RXH2 2/20 0.30
NPC1 O15118 2/20 0.30
MEN1 O00255 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Diphenylacetylene SCHEMBL619305 0.75 APP (0.60) TSHRAPPMAPTCYP1A2CYP3A4
Diphenylacetylene SCHEMBL339222 0.75 APP (0.60) TSHRAPPMAPTCYP1A2CYP3A4
SCHEMBL941489 0.71
Benzonitrile SCHEMBL30929383 0.69 TSHR (1.00) TSHRAPPMAOBMAOAMAPT
Benzonitrile SCHEMBL9464940 0.69 TSHR (1.00) TSHRAPPMAOBMAOAMAPT
Benzonitrile SCHEMBL27793280 0.69 TSHR (1.00) TSHRAPPMAOBMAOAMAPT
Benzonitrile SCHEMBL11044747 0.69
Benzonitrile SCHEMBL6640 0.69
Benzonitrile SCHEMBL21752925 0.69
Benzonitrile SCHEMBL27363057 0.69 TSHR (1.00) TSHRAPPMAOBMAOAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0907666-A1 PARTICLES COMPRISING AMPHIPHILIC COPOLYMERS, HAVING A CROSS-LINKED SHELL DOMAIN AND AN INTERIOR CORE DOMAIN, USEFUL FOR PHARMACEUTICAL AND OTHER APPLICATIONS G.D. Searle & Co. (US) 1999-04-14 EP disclosed
WO-1997049736-A2 PARTICLES COMPRISING AMPHIPHILIC COPOLYMERS, HAVING A CROSS-LINKED SHELL DOMAIN AND AN INTERIOR CORE DOMAIN, USEFUL FOR PHARMACEUTICAL AND OTHER APPLICATIONS G.D. SEARLE AND CO. (US) 1997-12-31 WO disclosed