SCHEMBL8386261

SCHEMBL8386261

CC(C)c1cc(-c2ccc(F)c3ccccc23)nc(NCCN)n1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1B P28222 1/20 0.64
HTR2B P41595 1/20 0.64
GPR65 Q8IYL9 1/20 0.64
KDM4E B2RXH2 6/20 0.41
ATM Q13315 1/20 0.38
NPSR1 Q6W5P4 2/20 0.37
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
BCDIN3D Q7Z5W3 2/20 0.35
SOS1 Q07889 1/20 0.35
PRKCH P24723 1/20 0.34
PRKCE Q02156 1/20 0.34
CAMK2D Q13557 1/20 0.34
CA12 O43570 1/20 0.34
CA3 P07451 1/20 0.34
CA4 P22748 1/20 0.34
CA6 P23280 1/20 0.34
CA5A P35218 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL5748951 0.91 HTR1B (0.54) HTR1BHTR2BGPR65KDM4EATM
Fumaric Acid SCHEMBL5748946 0.91 HTR1B (0.54) HTR1BHTR2BGPR65KDM4EATM
SCHEMBL5749566 0.91 HTR1B (0.60) HTR1BHTR2BGPR65KDM4EATM
SCHEMBL5749638 0.88 HTR1B (0.58) HTR1BHTR2BGPR65KDM4EATM
Bromide SCHEMBL8386216 0.88 HTR1B (0.58) HTR1BHTR2BGPR65KDM4EATM
Hydrochloric Acid SCHEMBL7132300 0.88 HTR1B (0.58) HTR1BHTR2BGPR65KDM4EATM
Hydrochloric Acid SCHEMBL5750473 0.88 HTR1B (0.58) HTR1BHTR2BGPR65KDM4EATM
SCHEMBL5750582 0.88 HTR1B (0.63) HTR1BHTR2BGPR65KDM4EATM
SCHEMBL5749037 0.87 HTR1B (0.57) HTR1BHTR2BGPR65KDM4EATM
Hydrochloric Acid SCHEMBL5772441 0.86 HTR1B (0.56) HTR1BHTR2BGPR65KDM4ESOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5958934-A 5-HT 2B ANTAGONIST SYNTEX (U.S.A.) INC. (US) 1999-09-28 US disclosed
US-5952331-A SELECTIVE 5HT2B ANTAGONISTS; SEROTONIN RECEPTOR ANTAGONIST; TREATING DISORDERS OF THE GASTROINTESTINAL TRACK, RESTENOSIS, ASTHMA AND OBSTRUCTIVE AIRWAY DISEASE, PROSTATIC HYPERPLASIA, GENERALIZED ANXIETY, PANIC DISORDER SYNTEX (USA) INC. (US) 1999-09-14 US disclosed
US-5863924-A Aryl pyrimidine derivatives SYNTEX (U.S.A.) INC. (US) 1999-01-26 US disclosed