SCHEMBL8395248

SCHEMBL8395248

CC(C)([NH])C(=O)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 7/20 0.54
SRC P12931 1/20 0.48
TSHR P16473 4/20 0.46
CES2 O00748 4/20 0.46
ALDH1A1 P00352 2/20 0.46
DAO P14920 1/20 0.46
NAPRT Q6XQN6 1/20 0.46
TDP1 Q9NUW8 4/20 0.45
HSD17B10 Q99714 2/20 0.45
MAPT P10636 3/20 0.42
POLB P06746 2/20 0.42
CYP3A4 P08684 2/20 0.42
CA2 P00918 2/20 0.42
CA4 P22748 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
PARP1 P09874 1/20 0.42
CYP2C19 P33261 1/20 0.42
RECQL P46063 1/20 0.42
BLM P54132 1/20 0.42
PMP22 Q01453 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6546660 0.83 CES1 (0.56) CES1SRCTSHRCES2ALDH1A1
SCHEMBL226691 0.80 CES1 (0.58) CES1SRCTSHRCES2ALDH1A1
SCHEMBL4618681 0.80 CES1 (0.58) CES1SRCTSHRCES2ALDH1A1
SCHEMBL21109870 0.80 CES1 (0.58) CES1SRCTSHRCES2ALDH1A1
SCHEMBL1606581 0.78 CES1 (0.56) CES1SRCTSHRCES2ALDH1A1
Hydrochloric Acid SCHEMBL2597972 0.78 CES1 (0.56) CES1SRCTSHRCES2ALDH1A1
SCHEMBL21310 0.78 CES1 (0.56) CES1SRCTSHRCES2ALDH1A1
SCHEMBL11341422 0.78 CES1 (0.56) CES1SRCTSHRCES2ALDH1A1
SCHEMBL9105008 0.78 CES1 (0.56) CES1SRCTSHRCES2ALDH1A1
SCHEMBL25930136 0.78 CES1 (0.56) CES1SRCTSHRCES2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5864043-A CARDIOVASCULAR DISORDERS AND ANGIOTENSIN ANTAGONIST KARL THOMAE GMBH (DE) 1999-01-26 US disclosed
US-5684029-A HYPOTENSIVE AGENTS KARL THOMAE GMBH (DE) 1997-11-04 US disclosed
US-5587393-A ANGIOTENSIN ANTAGONIST USEFUL IN TREATING HYPERTENSION DR. KARL THOMAE GMBH (DE) 1996-12-24 US disclosed
US-5541229-A ANGIOITENSIN II ANTAGONIST AS HYPOTENSIVE AGENTS, ANTIISCHEMIC AGENTS AND CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
US-5459147-A Angeotensin-antagonistic effects; hypotensive, antiischemic, and antidiabetic agents, treating glaucoma DR. KARL THOMAE GMBH (DE) 1995-10-17 US disclosed
US-5385925-A Benzimidazoles, pharmaceutical compositions containing these compounds and processes for preparing them DR. KARL THOMAE GMBH (DE) 1995-01-31 US disclosed