SCHEMBL8397204

SCHEMBL8397204

[CH2]NP(=O)(O)CCc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.56
CYP2D6 P10635 1/20 0.50
POLB P06746 1/20 0.49
CETP P11597 1/20 0.47
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
MMP1 P03956 1/20 0.47
MMP2 P08253 1/20 0.47
MMP3 P08254 1/20 0.47
CA9 Q16790 1/20 0.47
S1PR2 O95136 1/20 0.46
S1PR4 O95977 1/20 0.46
S1PR1 P21453 1/20 0.46
S1PR3 Q99500 1/20 0.46
MAPK1 P28482 1/20 0.45
ANPEP P15144 3/20 0.44
ERAP1 Q9NZ08 2/20 0.44
ERAP2 Q6P179 2/20 0.44
ACP3 P15309 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20626773 0.78 TSHR (0.62) TSHRCYP2D6POLBCETPCA12
SCHEMBL6030731 0.77 TSHR (0.88) TSHRCYP2D6POLBCETPCA12
SCHEMBL1101314 0.77 TSHR (0.67) TSHRCYP2D6POLBCETPCA12
SCHEMBL28543472 0.75 TSHR (0.64) TSHRCYP2D6POLBCETPCA12
SCHEMBL2517900 0.75 TSHR (0.84) TSHRCYP2D6POLBCETPCA12
SCHEMBL3874444 0.75 CYP2D6 (0.57) TSHRCYP2D6POLBCETPCA12
Phosphoric Acid SCHEMBL412030 0.74 TSHR (0.61) TSHRCYP2D6POLBCA12CA1
SCHEMBL3862229 0.74 TSHR (0.62) TSHRCYP2D6POLBCETPCA12
SCHEMBL28103039 0.74 TSHR (0.62) TSHRCYP2D6POLBCETPCA12
SCHEMBL11775231 0.74 TSHR (0.62) TSHRCYP2D6POLBCETPCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915704-A1 USE OF PHOSPHINYLOXYALKYL AND PHOSPHONAMIDOALKYL DERIVATIVES OF CYCLOPENTANE(ENE) AS THERAPEUTIC AGENTS Vision Pharmaceuticals L.P. (US) 1999-05-19 EP disclosed
WO-1997037666-A1 USE OF PHOSPHINYLOXYALKYL AND PHOSPHONAMIDOALKYL DERIVATIVES OF CYCLOPENTANE(ENE) AS THERAPEUTIC AGENTS ALLERGAN SALES, INC. (US) 1997-10-16 WO disclosed
US-5658897-A MUSCLE RELAXANTS AND OCULAR HYPOTENSIVE AGENTS ALLERGAN (US) 1997-08-19 US disclosed