SCHEMBL8400773

SCHEMBL8400773

CC1CC=C(c2nnn(C)n2)CN1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.36
PPARA Q07869 1/20 0.31
CHRM3 P20309 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8519257 0.80 CHRM2 (0.37) CHRM2
SCHEMBL8400243 0.74 CHRM2 (0.36) CHRM2CHRM3
SCHEMBL8400767 0.66 CHRM2 (0.37) CHRM2CHRM3
SCHEMBL8400245 0.63 CHRM2 (0.68) CHRM2CHRM3
SCHEMBL4790510 0.61 NISCH (0.39)
SCHEMBL46305 0.54 CCR1 (0.52) PPARA
SCHEMBL5844 0.54 SMN1; SMN2 (0.42) PPARA
SCHEMBL2644715 0.54 SMN1; SMN2 (0.46) PPARA
SCHEMBL23033807 0.54
SCHEMBL23576574 0.53 EPHX2 (0.41) PPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE36374-E 1,2,3-triazole and tetrazole substituted piperidine or tetrahydropyridine compounds useful as acetylcholine agonists H. LUNDBECK, A/S (DK) 1999-11-02 US disclosed
EP-0296721-B1 HETEROCYCLIC COMPOUNDS H. LUNDBECK A/S (DK) 1993-06-23 EP disclosed
US-4925858-A NERVOUS SYSTEM DISORDERS, ALZHEIMER*S DISEASE H. LUNDBECK A/S (DK) 1990-05-15 US disclosed
US-4866077-A TREATMENT OF NERVOUS SYSTEM DISORDERS SUCH AS ALZHEIMER*S DISEASE H. LUNDBECK A/S (DK) 1989-09-12 US disclosed
EP-0296721-A2 Heterocyclic compounds H. LUNDBECK A/S (DK) 1988-12-28 EP disclosed