SCHEMBL8407751

SCHEMBL8407751

Fc1ccc(COc2c(Cl)cc(OCC=C(Cl)Cl)cc2Cl)cc1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.42
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
MAOB P27338 10/20 0.38
MAOA P21397 1/20 0.38
APP P05067 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HTT P42858 1/20 0.38
NR4A2 P43354 2/20 0.38
NPSR1 Q6W5P4 1/20 0.37
PARP10 Q53GL7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8405583 0.89 MAPT (0.45) MAPTKMT2AMEN1MAOBMAOA
SCHEMBL8657189 0.88 PPARA (0.38) MAPTKMT2AMEN1MAOBMAOA
SCHEMBL8407693 0.86 MAOB (0.40) MAPTMAOBMAOAAPP
SCHEMBL8408601 0.86 KDM4E (0.41) MAPTKMT2AMEN1ALDH1A1NPSR1
SCHEMBL8405986 0.86 MAOB (0.44) MAOBMAOANR4A2PARP10
SCHEMBL8659980 0.86 PPARA (0.39) MAPTKMT2AMEN1MAOBMAOA
SCHEMBL8408840 0.86 MAOB (0.42) MAOBMAOA
SCHEMBL8408209 0.85 APP (0.40) MAPTMAOBAPPALDH1A1HTT
SCHEMBL8408873 0.85 IDO1 (0.41) MAPTMAOBMAOAALDH1A1
SCHEMBL8655532 0.85 FFAR1 (0.40) MAPTKMT2AMEN1MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5872137-A AROMATIC OXY DIHALOPRENE COMPOUNDS INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1999-02-16 US disclosed
EP-0722430-B1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL CO (JP) 1998-10-21 EP disclosed
EP-0722430-A1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1996-07-24 EP disclosed
WO-1996004228-A1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-02-15 WO disclosed