SCHEMBL8410995

SCHEMBL8410995

C=CCOc1ccc(CC(NC(C)=O)C(=O)Oc2ccccc2)cc1OCC=C

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 3/20 0.44
LMNA P02545 1/20 0.42
ALDH1A1 P00352 4/20 0.41
ADRB2 P07550 1/20 0.39
ADRB1 P08588 1/20 0.39
ADRB3 P13945 1/20 0.39
KMT2A Q03164 2/20 0.39
MAPT P10636 1/20 0.39
CASP1 P29466 1/20 0.39
PAM P19021 1/20 0.39
MEN1 O00255 1/20 0.39
CYP2D6 P10635 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
PPARG P37231 1/20 0.38
ITGB3 P05106 1/20 0.38
ITGA2B P08514 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27703700 0.78 TACR1 (0.61) TACR1ALDH1A1PAM
SCHEMBL26896456 0.77 TACR1 (0.47) TACR1ALDH1A1ADRB2ADRB1ADRB3
SCHEMBL20905743 0.77 TACR1 (0.47) TACR1ALDH1A1ADRB2ADRB1ADRB3
SCHEMBL11043757 0.76 TSHR (0.59) TACR1KMT2APAMITGB3ITGA2B
SCHEMBL11043759 0.76 TSHR (0.59) TACR1KMT2APAMITGB3ITGA2B
SCHEMBL2525910 0.76 TACR1 (0.43) TACR1LMNAALDH1A1KMT2AMAPT
SCHEMBL26896455 0.76 MME (0.51) TACR1ALDH1A1PPARGITGB3ITGA2B
SCHEMBL9493909 0.75 TACR1 (0.61) TACR1ALDH1A1CASP1PAM
SCHEMBL9493914 0.75 TACR1 (0.61) TACR1ALDH1A1CASP1PAM
SCHEMBL8409365 0.74 TACR1 (0.58) TACR1LMNAALDH1A1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5864041-A REACTING N-ACYL-3,4-DIHYDROXYPHENYLALAMINE DERIVATIVE WITH A HALOGEN RADICAL GENERATOR, A CERIUM SALT IN PRESENCE OR ABSENCE OF COPPER SALT CATALYST, OR A PERSULFATE SALT WITH COPPER CATALYST; USEFUL FOR TREATING NERVOUS SYSTEM DISORDERS SUMITOMO CHEMICAL COMPANY, LTD. (JP) 1999-01-26 US disclosed
US-5739387-A CATALYTIC CYCLIZATION WITH A CERIUM SALT OR A PERSULFATE SALT, DECYCLIZATION, DEBLOCKING AND DEPROTECTING SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-04-14 US disclosed