SCHEMBL8425012

SCHEMBL8425012

CCCC(=O)Nc1cnc[nH]1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH2 P25021 1/20 0.45
HRH1 P35367 1/20 0.45
HRH4 Q9H3N8 1/20 0.45
HRH3 Q9Y5N1 1/20 0.45
TP53 P04637 1/20 0.43
CYP2C19 P33261 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
GSK3B P49841 5/20 0.40
MAPK1 P28482 1/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
CCNA2 P20248 1/20 0.39
CDK2 P24941 1/20 0.39
CCNA1 P78396 1/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
MAPT P10636 1/20 0.39
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9954231 0.86 HRH2 (0.43) HRH2HRH1HRH4HRH3TP53
SCHEMBL18372644 0.81 HRH2 (0.41) HRH2HRH4HRH3CYP2C19MAPK1
SCHEMBL8818411 0.75 NPC1 (0.42) TP53POLBALDH1A1MAPTMEN1
SCHEMBL13743314 0.73 CYP3A4 (0.52) HRH2HRH1HRH4HRH3CYP2C19
SCHEMBL5518230 0.72
SCHEMBL14253913 0.71 HRH2 (0.42) HRH2HRH1HRH4HRH3TP53
SCHEMBL13033285 0.71 CYP3A4 (0.74) HRH2HRH1HRH4HRH3CYP2C19
SCHEMBL28522945 0.70 MAPK1 (0.49) TP53CYP2C19ADORA3ADORA2AADORA1
SCHEMBL13967999 0.70 HPGD (0.46) TP53CYP2C19GSK3BPOLBGAA
SCHEMBL13134161 0.70 JAK3 (0.42) TP53ALDH1A1HPGDMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5874501-A POLY(P-HYDROXYSTYRENE) WITH AROMATIC MOIETY AND ALIPHATIC MOIETY WITH INORGANIC OXIDE KEEHAN DONALD J (US) 1999-02-23 US disclosed
EP-0407554-B1 METALLIC OXIDE-OXIRANE POLYMERS AND PREPOLYMERS KEEHAN DONALD J (US) 1997-09-17 EP disclosed
US-5658996-A A LIQUID POLYEPOXIDE PREPOLYMER THE REACTION PRODUCT OF A TRISHYDROXYPHENYL, AN AROMATIC DIGLYCIDYL ETHER AND METAL OXIDE; CURABLE, LOW VISCOSITY; FORMED POLYEPOXIDE IS HEAT AND CHEMICAL RESISTANCE, ELONGATION, TOUGHNESS KEEHAN DONALD J (US) 1997-08-19 US disclosed
US-5169912-A Hydrolyzable oxygen bonding with epoxide; silica, titania; high performance coatings, adhesives KEEHAN DONALD J (US) 1992-12-08 US disclosed
US-5026816-A Reaction product of diglycidyl ether of (bisphenol a or resorcinol) with metallic oxide in presence of imidazole catalyst KEEHAN DONALD J (US) 1991-06-25 US disclosed