SCHEMBL8428129

SCHEMBL8428129

Cc1c(Cl)ccc2sccc12

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.42
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 3/20 0.40
GAA P10253 1/20 0.40
HTT P42858 1/20 0.40
CYP2A6 P11509 3/20 0.38
DYRK1A Q13627 1/20 0.32
NPC1 O15118 1/20 0.32
ICAM1 P05362 1/20 0.31
SELE P16581 1/20 0.31
VCAM1 P19320 1/20 0.31
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8404364 0.77 MAPT (0.44) MAPTKDM4EALDH1A1GAAHTT
SCHEMBL20563419 0.74 MAPT (0.42) MAPTKDM4EALDH1A1GAAHTT
SCHEMBL2056250 0.74 MAPT (0.42) MAPTKDM4EALDH1A1GAAHTT
SCHEMBL9394238 0.74 KDM4E (0.42) MAPTKDM4EALDH1A1GAAHTT
SCHEMBL18069886 0.74 MAPT (0.42) MAPTKDM4EALDH1A1GAAHTT
SCHEMBL18876006 0.74 CYP2A6 (0.42) MAPTKDM4EALDH1A1GAAHTT
SCHEMBL2498909 0.72 KDM4E (0.45) MAPTKDM4EALDH1A1GAAHTT
SCHEMBL29352476 0.72 KDM4E (0.45) MAPTKDM4EALDH1A1GAAHTT
SCHEMBL22504295 0.72 KDM4E (0.42) MAPTKDM4EALDH1A1GAAHTT
SCHEMBL24344559 0.71 KDM4E (0.40) MAPTKDM4EALDH1A1GAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5922733-A ADMINISTERING TO TREAT CENTRAL NERVOUS SYSTEM DISORDERS SUCH AS ANXIETY, DEPRESSION, EPILEPSY, OBSESSIVE COMPULSIVE DISORDERS, ANOREXIA, BULIMIA AND ALZHEIMER'S DISEASE SMITHKLINE BEECHAM P.L.C. (GB) 1999-07-13 US disclosed
EP-0770076-A1 BENZOCONDENSED FIVE MEMBERED HETEROCYCLE CARBOXAMIDES AS 5HT2B/2C RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1997-05-02 EP disclosed
WO-1996002537-A1 BENZOCONDENSED FIVE MEMBERED HETEROCYCLE CARBOXAMIDES AS 5HT2B/2C RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1996-02-01 WO disclosed