SCHEMBL8428518

SCHEMBL8428518

CN(C)CCCOc1ccc(C=c2[nH]c(=O)c(=Cc3ccc(C(=O)N4CCc5ccccc5C4)cc3)[nH]c2=O)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 3/20 0.52
HSP90B1 P14625 2/20 0.49
TRAP1 Q12931 2/20 0.49
SERPINE1 P05121 2/20 0.48
HPGD P15428 4/20 0.47
MAPT P10636 2/20 0.47
LMNA P02545 1/20 0.47
HRH3 Q9Y5N1 1/20 0.46
MTHFD1 P11586 1/20 0.45
MTHFD2 P13995 1/20 0.45
ALDH1A1 P00352 1/20 0.45
TSHR P16473 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HSD17B10 Q99714 1/20 0.45
TP53 P04637 1/20 0.44
MEN1 O00255 1/20 0.43
HTT P42858 1/20 0.43
RECQL P46063 1/20 0.43
KMT2A Q03164 1/20 0.43
CACNA1H O95180 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8428514 1.00 CACNA1B (0.52) CACNA1BHSP90B1TRAP1SERPINE1HPGD
SCHEMBL8424360 0.83 PRMT5 (0.46) CACNA1BSERPINE1HPGDMAPTLMNA
SCHEMBL8424366 0.83 PRMT5 (0.46) CACNA1BSERPINE1HPGDMAPTLMNA
SCHEMBL8428423 0.82 DRD3 (0.53) CACNA1BHPGDLMNAHRH3
SCHEMBL8428415 0.82 DRD3 (0.53) CACNA1BHPGDLMNAHRH3
SCHEMBL6378369 0.78 SERPINE1 (0.67) SERPINE1HRH3
SCHEMBL8494225 0.78 SERPINE1 (0.67) SERPINE1HRH3
SCHEMBL8495273 0.78 SERPINE1 (0.59) SERPINE1HRH3ALDH1A1SMN1; SMN2
SCHEMBL8495305 0.78 SERPINE1 (0.59) SERPINE1HRH3ALDH1A1SMN1; SMN2
SCHEMBL8492151 0.77 SERPINE1 (0.55) SERPINE1HRH3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0745070-A1 PHARMACEUTICAL PIPERAZINE COMPOUNDS XENOVA LIMITED (GB) 1996-12-04 EP claimed
WO-1995021832-A1 PHARMACEUTICAL PIPERAZINE COMPOUNDS XENOVA LIMITED (GB) 1995-08-17 WO claimed
US-5891877-A INHIBITORS OF PLASMINOGEN ACTIVATOR INHIBITOR XENOVA LIMITED (GB) 1999-04-06 US disclosed
EP-0745070-A1 PHARMACEUTICAL PIPERAZINE COMPOUNDS XENOVA LIMITED (GB) 1996-12-04 EP disclosed
WO-1995021832-A1 PHARMACEUTICAL PIPERAZINE COMPOUNDS XENOVA LIMITED (GB) 1995-08-17 WO disclosed