SCHEMBL8439563

SCHEMBL8439563

Cc1ccc(CN2CCN(C(=O)c3c[nH]c4ccccc34)CC2)cc1

nearest known ligand 0.82

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 2/20 0.82
HTT P42858 2/20 0.82
HDAC1 Q13547 4/20 0.73
HDAC6 Q9UBN7 4/20 0.73
ALDH1A1 P00352 2/20 0.61
KMT2A Q03164 2/20 0.61
MAPT P10636 1/20 0.61
GFER P55789 1/20 0.58
HDAC3 O15379 1/20 0.58
HDAC2 Q92769 1/20 0.58
DRD2 P14416 1/20 0.57
DRD3 P35462 1/20 0.57
TP53 P04637 1/20 0.57
HRH3 Q9Y5N1 2/20 0.55
LMNA P02545 2/20 0.55
SMN1; SMN2 Q16637 1/20 0.53
IGF1R P08069 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8301611 0.90 MAPK14 (1.00) MAPK14HTTHDAC1HDAC6ALDH1A1
SCHEMBL8445048 0.88 MAPK14 (0.82) MAPK14HTTHDAC1HDAC6ALDH1A1
SCHEMBL8436827 0.86 MAPK14 (0.75) MAPK14HTTHDAC1HDAC6ALDH1A1
SCHEMBL8303336 0.86 MAPK14 (0.82) MAPK14HTTHDAC1HDAC6ALDH1A1
SCHEMBL12918551 0.85 MAPK14 (0.77) MAPK14HTTHDAC1HDAC6ALDH1A1
SCHEMBL24358707 0.82 GFER (0.81) MAPK14HTTHDAC1HDAC6ALDH1A1
SCHEMBL16599095 0.81 RGS12 (0.78) MAPK14HTTHDAC1HDAC6ALDH1A1
SCHEMBL29335990 0.80 MAPK14 (0.73) MAPK14HTTHDAC1HDAC6ALDH1A1
SCHEMBL16598785 0.79 MAPK14 (0.78) MAPK14HTTHDAC1HDAC6ALDH1A1
SCHEMBL948677 0.79 GFER (0.71) MAPK14HTTHDAC1HDAC6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0922042-A1 NOVEL PIPERAZINE CONTAINING COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1999-06-16 EP disclosed
WO-1998006715-A1 NOVEL PIPERAZINE CONTAINING COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1998-02-19 WO disclosed