SCHEMBL8444592

SCHEMBL8444592

COc1ccc(-n2cnnn2)cc1C(=O)N1CCC(CCN2CCC(C(=O)NO)(c3ccccc3)CC2)(c2ccc(C)c(C)c2)C1

nearest known ligand 0.54

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TACR2 P21452 9/20 0.54
TACR1 P25103 9/20 0.54
TACR3 P29371 1/20 0.49
HRH1 P35367 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8446075 0.95 TACR2 (0.56) TACR2TACR1TACR3HRH1
SCHEMBL8441021 0.94 TACR2 (0.47) TACR2TACR1TACR3HRH1
SCHEMBL8438789 0.94 TACR2 (0.55) TACR2TACR1TACR3HRH1
SCHEMBL8441824 0.93 TACR2 (0.47) TACR2TACR1TACR3HRH1
SCHEMBL8435623 0.92 TACR2 (0.65) TACR2TACR1TACR3HRH1
SCHEMBL8441186 0.92 TACR2 (0.65) TACR2TACR1TACR3HRH1
SCHEMBL8439962 0.92 TACR2 (0.65) TACR2TACR1TACR3HRH1
SCHEMBL8434741 0.92 TACR2 (0.47) TACR2TACR1TACR3HRH1
SCHEMBL8442938 0.92 TACR2 (0.53) TACR2TACR1TACR3HRH1
SCHEMBL8444744 0.92 TACR2 (0.54) TACR2TACR1TACR3HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946548-A1 NOVEL HETEROCYCLIC SUBSTITUTED PYRROLIDINE AMIDE DERIVATIVES HOECHST MARION ROUSSEL, INC. (US) 1999-10-06 EP disclosed
WO-1998027086-A1 NOVEL HETEROCYCLIC SUBSTITUTED PYRROLIDINE AMIDE DERIVATIVES HOECHST MARION ROUSSEL, INC. (US) 1998-06-25 WO disclosed