SCHEMBL8458513

SCHEMBL8458513

CCOC(=O)c1ccc(C=C(C)c2ccc3c(c2)CCC(=O)CC3)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.43
HPGD P15428 2/20 0.43
RARB P10826 6/20 0.43
RARG P13631 6/20 0.43
RARA P10276 5/20 0.43
SRD5A1 P18405 1/20 0.42
SRD5A2 P31213 1/20 0.42
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA7 P43166 2/20 0.41
CA9 Q16790 2/20 0.41
CA14 Q9ULX7 2/20 0.41
ESR1 P03372 1/20 0.41
ESR2 Q92731 1/20 0.41
ALDH1A1 P00352 3/20 0.41
NPSR1 Q6W5P4 2/20 0.41
HSP90AA1 P07900 1/20 0.41
CACNA1B Q00975 1/20 0.41
APBA1 Q02410 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8458507 1.00 HTT (0.43) HTTHPGDRARBRARGRARA
SCHEMBL9419049 0.89 HPGD (0.44) HTTHPGDRARBRARGRARA
SCHEMBL9419050 0.89 HPGD (0.44) HTTHPGDRARBRARGRARA
SCHEMBL9863478 0.86 RARG (0.55) RARBRARGRARAALDH1A1NPSR1
SCHEMBL9863485 0.86 RARG (0.55) RARBRARGRARAALDH1A1NPSR1
SCHEMBL9419019 0.86 RARB (0.48) HTTHPGDRARBRARGRARA
SCHEMBL9418999 0.86 RARB (0.46) HTTHPGDRARBRARGRARA
SCHEMBL7223039 0.86 RARB (0.48) HTTHPGDRARBRARGRARA
SCHEMBL8460900 0.86 DRD3 (0.44) HTTHPGDRARBRARGRARA
SCHEMBL9418995 0.86 RARB (0.46) HTTHPGDRARBRARGRARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0315071-B1 Benzocyclohepten derivatives, their preparation and utilisation for pharmaceutics HOFFMANN LA ROCHE (CH) 1994-07-20 EP claimed
WO-1999048529-A1 RETINOID-GLITAZONE COMBINATIONS WARNER-LAMBERT COMPANY (US) 1999-09-30 WO disclosed
EP-0808159-A1 USE OR RETINOIDS TO LOWER PLASMA LEVELS OF LIPOPROTEIN (a) WARNER-LAMBERT COMPANY (US) 1997-11-26 EP disclosed
WO-1996024344-A1 USE OF RETINOIDS TO LOWER PLASMA LEVELS OF LIPOPROTEIN (a) WARNER-LAMBERT COMPANY (US) 1996-08-15 WO disclosed
US-5489611-A ADMINISTERING A RETINOID COMPOUND WARNER-LAMBERT COMPANY (US) 1996-02-06 US disclosed
US-4992574-A Skin disorders, antiallergens, antiinflammatory agent HOFFMANN-LA ROCHE INC. (US) 1991-02-12 US disclosed