SCHEMBL8458989

SCHEMBL8458989

NCCNCCc1ccccn1

nearest known ligand 0.66

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 2/20 0.66
CYP1A2 P05177 3/20 0.60
ALDH1A1 P00352 2/20 0.60
CYP2C19 P33261 1/20 0.60
HRH3 Q9Y5N1 1/20 0.59
LMNA P02545 2/20 0.58
TAAR1 Q96RJ0 1/20 0.58
ALOX15 P16050 1/20 0.58
CHRM2 P08172 1/20 0.56
CYP2D6 P10635 1/20 0.54
TDP1 Q9NUW8 1/20 0.50
DPP7 Q9UHL4 1/20 0.50
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4397357 0.93 HRH1 (0.64) HRH1CYP1A2ALDH1A1CYP2C19HRH3
SCHEMBL1921574 0.90 HRH3 (0.70) HRH1CYP1A2ALDH1A1CYP2C19HRH3
SCHEMBL23053146 0.88 CYP1A2 (0.69) HRH1CYP1A2ALDH1A1CYP2C19HRH3
SCHEMBL28455774 0.84 CHRM2 (0.74) HRH1CYP1A2ALDH1A1HRH3LMNA
SCHEMBL3319194 0.84 CHRM2 (0.74) HRH1CYP1A2ALDH1A1HRH3LMNA
SCHEMBL160154 0.83 CHRM2 (0.73) HRH1CYP1A2ALDH1A1HRH3LMNA
SCHEMBL5707525 0.82 CYP1A2 (0.61) HRH1CYP1A2ALDH1A1CYP2C19HRH3
SCHEMBL6890029 0.82 CHRM2 (0.57) HRH1CYP1A2ALDH1A1CYP2C19HRH3
SCHEMBL5707323 0.81 CYP1A2 (0.60) HRH1CYP1A2ALDH1A1CYP2C19HRH3
SCHEMBL10931346 0.81 CYP1A2 (0.60) HRH1CYP1A2ALDH1A1CYP2C19HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999039575-A2 SYNERGISTIC BIOCIDAL ACTIVITY OF TERNARY COMPLEXES OF NEGATIVELY -CHARGED BIOCIDES (COMPONENT A), TRANSITION METAL IONS (COMPONENT B), AND NEUTRAL CHELATORS (COMPONENT C) YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 1999-08-12 WO claimed
JP-60123508-A None JP disclosed
JP-59030802-A None JP disclosed
JP-S60123508-A PRODUCTION OF PYRIDYLALKYLAMINOPOLYCARBOXYLIC ACID TYPE CHELATE RESIN AGENCY OF IND SCIENCE & TECHNOL 1985-07-02 JP disclosed
JP-S5930802-A PREPARATION OF CHELATE RESIN HAVING PYRIDYLALKYLAMINE AND PYRIDYLALKYLAMINOPOLYCARBOXYLIC ACID AS LIGAND AGENCY OF IND SCIENCE & TECHNOL 1984-02-18 JP disclosed